SCHEMBL8713259

SCHEMBL8713259

COc1ccc(OC)c(N(CCN2CCC(C(=O)c3ccc(F)cc3)CC2)C(=O)c2ccc(NC(C)=O)cc2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 3/20 0.51
CYP2C9 P11712 2/20 0.51
CYP1A2 P05177 1/20 0.51
GAA P10253 1/20 0.51
SMN1; SMN2 Q16637 4/20 0.50
LMNA P02545 3/20 0.50
ALDH1A1 P00352 3/20 0.50
HTT P42858 2/20 0.50
GLA P06280 1/20 0.50
MAPK1 P28482 1/20 0.50
HSD11B1 P28845 3/20 0.48
MAPT P10636 1/20 0.47
CYP2D6 P10635 1/20 0.47
POLB P06746 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
DRD2 P14416 1/20 0.45
HTR2A P28223 1/20 0.45
HTR2C P28335 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL8713807 0.96 CYP2C19 (0.47) CYP2C19CYP2C9CYP1A2GAASMN1; SMN2
Fumaric Acid SCHEMBL8713808 0.96 CYP2C19 (0.47) CYP2C19CYP2C9CYP1A2GAASMN1; SMN2
SCHEMBL8710763 0.94 CYP2C19 (0.51) CYP2C19CYP2C9CYP1A2GAASMN1; SMN2
SCHEMBL8713319 0.90 CYP2C19 (0.54) CYP2C19CYP2C9CYP1A2GAASMN1; SMN2
Fumaric Acid SCHEMBL8712465 0.90 CYP2C19 (0.47) CYP2C19CYP2C9CYP1A2GAASMN1; SMN2
Fumaric Acid SCHEMBL8712464 0.90 CYP2C19 (0.47) CYP2C19CYP2C9CYP1A2GAASMN1; SMN2
SCHEMBL8716522 0.89 ALDH1A1 (0.53) CYP2C19SMN1; SMN2LMNAALDH1A1HTT
Oxalic Acid SCHEMBL8711790 0.88 CYP2C19 (0.51) CYP2C19CYP2C9CYP1A2GAASMN1; SMN2
SCHEMBL8712161 0.88 CYP2C9 (0.58) CYP2C19CYP2C9CYP1A2GAASMN1; SMN2
SCHEMBL8711355 0.86 HSD11B1 (0.51) CYP2C19CYP2C9CYP1A2GAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5728835-A HYPOTENSIVE AGENTS; ANTIISCHEMIC AGENTS TOA EIYO, LTD. (JP) 1998-03-17 US disclosed
EP-0661266-A1 Substituted cyclic amine compounds as 5HT2 antagonists TOA EIYO LTD. (JP) 1995-07-05 EP disclosed