SCHEMBL8713323

SCHEMBL8713323

O=C(Cl)c1nn(C2CCCC2)c2ccccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 9/20 0.45
HTR3E A5X5Y0 1/20 0.45
SLC22A2 O15244 1/20 0.45
HTR3B O95264 1/20 0.45
CHRNB2 P17787 1/20 0.45
CHRNA3 P32297 1/20 0.45
CHRNA4 P43681 1/20 0.45
KCNH2 Q12809 1/20 0.45
HTR3D Q70Z44 1/20 0.45
HTR3C Q8WXA8 1/20 0.45
SLC47A1 Q96FL8 1/20 0.45
PDE4A P27815 2/20 0.42
PDE4B Q07343 2/20 0.42
PDE4C Q08493 2/20 0.42
PDE4D Q08499 2/20 0.42
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42
ALDH1A1 P00352 2/20 0.41
CYP3A4 P08684 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8718851 0.99 HTR3A (0.44) HTR3AHTR3ESLC22A2HTR3BCHRNB2
SCHEMBL8717365 0.97 HTR3A (0.48) HTR3AHTR3ESLC22A2HTR3BCHRNB2
SCHEMBL3411552 0.87 KDM4E (0.47) HTR3AHTR3ESLC22A2HTR3BCHRNB2
SCHEMBL8876610 0.85 ELANE (0.51) HTR3AHTR3ESLC22A2HTR3BCHRNB2
SCHEMBL8718634 0.85 KDM4E (0.49) HTR3AHTR3ESLC22A2HTR3BCHRNB2
SCHEMBL2078485 0.84 HTR3A (0.46) HTR3AHTR3ESLC22A2HTR3BCHRNB2
SCHEMBL21725181 0.82 ELANE (0.54) HTR3AHTR3ESLC22A2HTR3BCHRNB2
SCHEMBL719399 0.81 ELANE (0.53) HTR3AHTR3ESLC22A2HTR3BCHRNB2
SCHEMBL31429395 0.80 CYP3A4 (0.44) HTR3AHTR3ESLC22A2HTR3BCHRNB2
SCHEMBL2077051 0.79 ELANE (0.54) HTR3AHTR3ESLC22A2HTR3BCHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0708105-B1 5-HT4 receptor agonists NISSHIN FLOUR MILLING CO (JP) 1998-12-23 EP disclosed
US-5684003-A GASTROINTESTINAL DISORDERS OR ANTIULCER AGENTS NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-11-04 US disclosed
EP-0708105-A1 5-HT4 receptor agonists NISSHIN FLOUR MILLING CO., LTD. (JP) 1996-04-24 EP disclosed