SCHEMBL8713374

SCHEMBL8713374

Cc1c(C)c([N+](=O)[O-])c(C)c2c1OC(C)(C)C2c1cccnc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
GSK3A P49840 1/20 0.33
GSK3B P49841 1/20 0.33
TNKS O95271 1/20 0.33
ALDH1A1 P00352 4/20 0.33
KDM4E B2RXH2 3/20 0.33
MAPT P10636 2/20 0.33
LMNA P02545 2/20 0.33
G6PD P11413 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
RAB9A P51151 1/20 0.33
GLA P06280 1/20 0.32
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32
CASP1 P29466 1/20 0.32
CASP7 P55210 1/20 0.32
HSD17B10 Q99714 1/20 0.32
MAPK1 P28482 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8712974 0.86 ALDH1A1 (0.34) MEN1KMT2AALDH1A1MAPTLMNA
SCHEMBL9665303 0.81 CYP2A6 (0.35) GSK3AGSK3BTNKSALDH1A1KDM4E
SCHEMBL8718473 0.81 ACHE (0.37) MEN1KMT2AALDH1A1MAPTLMNA
Hydrochloric Acid SCHEMBL9668091 0.80 CYP2A6 (0.34) GSK3AGSK3BTNKSALDH1A1KDM4E
SCHEMBL8713506 0.80 CYP2A6 (0.34) GSK3AGSK3BTNKSALDH1A1KDM4E
SCHEMBL8716319 0.79 NPSR1 (0.36) ALDH1A1L3MBTL1HTT
SCHEMBL8715950 0.76 TSHR (0.35) GSK3AGSK3BTNKSMAPTRAB9A
SCHEMBL8716496 0.73 ALDH1A1 (0.38) KMT2AALDH1A1KDM4EMAPTLMNA
SCHEMBL8714404 0.73 KCNH2 (0.39)
SCHEMBL5348524 0.68 MAPT (0.38) MEN1KMT2AALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5770772-A 4-FORMYLAMINO-2,3,5-TRIMETHYL-1-(2-METHYL-2-PROPENYLOXY) -BENZENE; ARTERIOSCLEROSIS, BRAIN AND CARDIOVASCULAR DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-06-23 US disclosed
US-5594154-A 5-AMINO-2-BROMOMETHYL-2,4,6,7-TETRAMETHYL-2,3-DIHYDROBENZO(B) FURANS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-01-14 US disclosed
US-5478844-A Method of using aminocoumaran derivatives for treating cerebrovascular diseases TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-12-26 US disclosed
EP-0483772-B1 Aminocoumaran derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-09-13 EP disclosed
US-5376681-A Aminocoumaran derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-12-27 US disclosed
EP-0483772-A1 Aminocoumaran derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-05-06 EP disclosed