SCHEMBL8713816

SCHEMBL8713816

CCCn1c(=O)c2c(nc(C)n2CCc2ccc(OCc3ccccc3)cc2)n(CCC)c1=O

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 6/20 0.50
ADORA3 P0DMS8 5/20 0.50
TSHR P16473 1/20 0.49
HSD17B10 Q99714 1/20 0.49
ADORA2A P29274 5/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
ADORA1 P30542 3/20 0.47
GFER P55789 1/20 0.47
POLB P06746 1/20 0.47
MAPT P10636 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8710110 0.82 ADORA2B (0.61) ADORA2BADORA3TSHRHSD17B10ADORA2A
SCHEMBL1946830 0.82 ADORA2B (0.62) ADORA2BADORA3ADORA2AADORA1MAPT
SCHEMBL3226126 0.77 ADORA1 (0.60) ADORA2BADORA3ADORA2AADORA1
SCHEMBL1061950 0.76 ADORA2A (0.53) ADORA2BADORA3ADORA2AADORA1
SCHEMBL1945104 0.76 ADORA2B (0.52) ADORA2BADORA3ADORA2AADORA1
SCHEMBL12245132 0.72 ADORA2A (0.55) ADORA2BADORA3ADORA2AADORA1MAPT
SCHEMBL1065789 0.72 ADORA2B (0.73) ADORA2BADORA3HSD17B10ADORA2AMEN1
SCHEMBL1947373 0.72 ADORA2B (0.52) ADORA2BADORA3ADORA2AADORA1
SCHEMBL8578138 0.72 ADORA3 (0.56) ADORA2BADORA3ADORA2AKMT2AADORA1
SCHEMBL9708336 0.71 ADORA3 (0.46) ADORA2BADORA3ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5840729-A ATTENUATING COGNITIVE DEFICIT MERRELL PHARMACEUTICALS INC. (US) 1998-11-24 US disclosed