SCHEMBL8713978

SCHEMBL8713978

Cc1c(C)c2c(c(C)c1NS(C)(=O)=O)CC(C)(C)O2

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8716244 0.80 ALDH1A1 (0.51) ALDH1A1SMN1; SMN2LMNAHTTCYP1A2
SCHEMBL29455782 0.78 ALDH1A1 (0.32) ALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL8713217 0.77 ALDH1A1 (0.31) ALDH1A1SMN1; SMN2HSP90AA1HSP90AB1
SCHEMBL8714063 0.76 ALDH1A1 (0.32) ALDH1A1SMN1; SMN2
SCHEMBL12811732 0.76 HSP90AA1 (0.38) ALDH1A1SMN1; SMN2LMNAHTTCYP1A2
SCHEMBL8716967 0.75 MEN1 (0.36) ALDH1A1SMN1; SMN2LMNACYP1A2CYP3A4
SCHEMBL4047614 0.74 HSP90AA1 (0.37) ALDH1A1SMN1; SMN2LMNAHTTCYP1A2
SCHEMBL29561615 0.74 HSP90AA1 (0.37) ALDH1A1SMN1; SMN2LMNAHTTCYP1A2
SCHEMBL8747110 0.73 ALDH1A1 (0.33) ALDH1A1SMN1; SMN2LMNAHTTCYP1A2
Hydrochloric Acid SCHEMBL8717770 0.73 EZH2 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5770772-A 4-FORMYLAMINO-2,3,5-TRIMETHYL-1-(2-METHYL-2-PROPENYLOXY) -BENZENE; ARTERIOSCLEROSIS, BRAIN AND CARDIOVASCULAR DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-06-23 US disclosed
US-5594154-A 5-AMINO-2-BROMOMETHYL-2,4,6,7-TETRAMETHYL-2,3-DIHYDROBENZO(B) FURANS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-01-14 US disclosed
US-5478844-A Method of using aminocoumaran derivatives for treating cerebrovascular diseases TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-12-26 US disclosed
EP-0483772-B1 Aminocoumaran derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-09-13 EP disclosed
US-5376681-A Aminocoumaran derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-12-27 US disclosed
CN-1071165-A Aminocoumaran derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1993-04-21 CN disclosed
EP-0483772-A1 Aminocoumaran derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-05-06 EP disclosed