SCHEMBL8716244

SCHEMBL8716244

Cc1ccc(S(=O)(=O)Nc2c(C)c(C)c3c(c2C)CC(C)(C)O3)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
LMNA P02545 3/20 0.47
HTT P42858 2/20 0.47
CYP26A1 O43174 1/20 0.44
CYP26B1 Q9NR63 1/20 0.44
FFAR4 Q5NUL3 1/20 0.43
EDNRB P24530 1/20 0.41
EDNRA P25101 1/20 0.41
CYTH2 Q99418 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
CYP2C19 P33261 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
KDM4E B2RXH2 1/20 0.39
BRD4 O60885 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8713217 0.70 ALDH1A1 (0.31) ALDH1A1SMN1; SMN2
SCHEMBL8714063 0.70 ALDH1A1 (0.32) ALDH1A1SMN1; SMN2
SCHEMBL2371862 0.69 HSP90AA1 (0.42) ALDH1A1SMN1; SMN2LMNAHTTCYP2C19
SCHEMBL8716967 0.69 MEN1 (0.36) ALDH1A1SMN1; SMN2LMNACYP1A2CYP3A4
SCHEMBL13183198 0.68 RAPGEF4 (0.42) ALDH1A1SMN1; SMN2LMNAHTTEDNRA
SCHEMBL4047614 0.68 HSP90AA1 (0.37) ALDH1A1SMN1; SMN2LMNAHTTCYP2C19
SCHEMBL8720009 0.68 MAPT (0.44) ALDH1A1SMN1; SMN2LMNAHTTKDM4E
Hydrochloric Acid SCHEMBL8717770 0.67 EZH2 (0.30)
SCHEMBL12811732 0.66 HSP90AA1 (0.38) ALDH1A1SMN1; SMN2LMNAHTTCYP2C19
SCHEMBL8718408 0.66 MEN1 (0.39) ALDH1A1SMN1; SMN2LMNACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5770772-A 4-FORMYLAMINO-2,3,5-TRIMETHYL-1-(2-METHYL-2-PROPENYLOXY) -BENZENE; ARTERIOSCLEROSIS, BRAIN AND CARDIOVASCULAR DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-06-23 US disclosed
US-5594154-A 5-AMINO-2-BROMOMETHYL-2,4,6,7-TETRAMETHYL-2,3-DIHYDROBENZO(B) FURANS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-01-14 US disclosed
US-5478844-A Method of using aminocoumaran derivatives for treating cerebrovascular diseases TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-12-26 US disclosed
EP-0483772-B1 Aminocoumaran derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-09-13 EP disclosed
US-5376681-A Aminocoumaran derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-12-27 US disclosed
EP-0483772-A1 Aminocoumaran derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-05-06 EP disclosed