SCHEMBL8714004

SCHEMBL8714004

c1ccc2c(N3CC[N]CC3)n[nH]c2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.44
KDM4E B2RXH2 2/20 0.44
GAA P10253 2/20 0.44
PDPK1 O15530 1/20 0.44
CYP3A4 P08684 1/20 0.44
HPGD P15428 2/20 0.42
ALDH1A1 P00352 1/20 0.42
ALPL P05186 1/20 0.42
IDO1 P14902 1/20 0.42
TTK P33981 1/20 0.42
MAPK10 P53779 1/20 0.42
TNKS O95271 2/20 0.41
PARP2 Q9UGN5 2/20 0.41
CYP1A2 P05177 1/20 0.39
LRRK2 Q5S007 3/20 0.38
CDC7 O00311 2/20 0.38
ADRA2A P08913 2/20 0.38
ENPP1 P22413 1/20 0.38
PIM1 P11309 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3067812 0.86 HPGD (0.55) PARP1KDM4EGAAPDPK1CYP3A4
SCHEMBL18228562 0.86 HPGD (0.55) PARP1KDM4EGAAPDPK1CYP3A4
SCHEMBL4053256 0.84 HPGD (0.58) PARP1KDM4EGAAPDPK1CYP3A4
SCHEMBL29468202 0.83 KDM4E (0.54) PARP1KDM4EGAAPDPK1CYP3A4
SCHEMBL1132419 0.83 KDM4E (0.54) PARP1KDM4EGAAPDPK1CYP3A4
SCHEMBL23536581 0.81 LRRK2 (0.56) KDM4EGAAHPGDALDH1A1MAPK10
SCHEMBL1545498 0.81 CDC7 (0.53) PARP1KDM4EALDH1A1MAPK10CDC7
Hydrochloric Acid SCHEMBL5767318 0.81 KDM4E (0.56) PARP1KDM4EGAAPDPK1CYP3A4
SCHEMBL9778335 0.79 KMT2A (0.50) PARP1CYP3A4HPGDALDH1A1TNKS
SCHEMBL23570187 0.79 MAPK1 (0.44) PARP1KDM4EGAAPDPK1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5854263-A 1- (1,4-benzodioxanyl)alkyl!-3-(heteroaryl) pyrrolidines and related compounds and their therapeutic utility HOECHST MARION ROUSSEL, INC. (US) 1998-12-29 US disclosed