SCHEMBL8714385

SCHEMBL8714385

COc1cccc(N(CCN2CCC(C(=O)c3ccc(F)cc3)CC2)C(=O)c2ccc(NC(C)=O)c(OC)c2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.51
CYP2D6 P10635 1/20 0.51
HSD11B1 P28845 4/20 0.49
HSD17B10 Q99714 1/20 0.47
ALDH1A1 P00352 2/20 0.45
LMNA P02545 2/20 0.45
HTT P42858 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
KMT2A Q03164 3/20 0.44
MEN1 O00255 1/20 0.44
UBE2N P61088 1/20 0.44
MAPT P10636 1/20 0.44
WNT3A P56704 1/20 0.42
TNKS2 Q9H2K2 1/20 0.42
HTR2A P28223 3/20 0.42
HTR2C P28335 2/20 0.42
DRD2 P14416 1/20 0.42
CYP1A2 P05177 1/20 0.42
GAA P10253 1/20 0.42
CYP2C9 P11712 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8715758 0.93 HSD11B1 (0.48) CYP2C19CYP2D6HSD11B1HSD17B10ALDH1A1
SCHEMBL8715019 0.91 CYP2C19 (0.51) CYP2C19CYP2D6HSD11B1HSD17B10ALDH1A1
SCHEMBL8710891 0.90 HSD11B1 (0.51) CYP2C19CYP2D6HSD11B1LMNASMN1; SMN2
SCHEMBL8711355 0.90 HSD11B1 (0.51) CYP2C19CYP2D6HSD11B1ALDH1A1LMNA
SCHEMBL8712025 0.89 CYP2D6 (0.49) CYP2C19CYP2D6HSD11B1HSD17B10ALDH1A1
Hydrochloric Acid SCHEMBL8711024 0.89 HSD11B1 (0.50) CYP2C19CYP2D6HSD11B1ALDH1A1LMNA
SCHEMBL8714991 0.88 HSD11B1 (0.51) CYP2C19CYP2D6HSD11B1ALDH1A1LMNA
Fumaric Acid SCHEMBL8714787 0.87 CYP2C19 (0.47) CYP2C19CYP2D6HSD11B1HSD17B10ALDH1A1
Fumaric Acid SCHEMBL8714788 0.87 CYP2C19 (0.47) CYP2C19CYP2D6HSD11B1HSD17B10ALDH1A1
Fumaric Acid SCHEMBL8716648 0.86 HSD11B1 (0.47) CYP2C19CYP2D6HSD11B1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5728835-A HYPOTENSIVE AGENTS; ANTIISCHEMIC AGENTS TOA EIYO, LTD. (JP) 1998-03-17 US disclosed
EP-0661266-A1 Substituted cyclic amine compounds as 5HT2 antagonists TOA EIYO LTD. (JP) 1995-07-05 EP disclosed