SCHEMBL8715019

SCHEMBL8715019

COc1ccc(N(CCN2CCC(C(=O)c3ccc(F)cc3)CC2)C(=O)c2ccc(NC(C)=O)c(OC)c2)cc1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.51
CYP2D6 P10635 1/20 0.51
OPRM1 P35372 1/20 0.49
CYP1A2 P05177 1/20 0.48
GAA P10253 1/20 0.48
CYP2C9 P11712 1/20 0.48
PTGIR P43119 1/20 0.47
HSD17B10 Q99714 1/20 0.47
ALDH1A1 P00352 2/20 0.47
LMNA P02545 2/20 0.47
HSD11B1 P28845 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
KMT2A Q03164 1/20 0.47
HTT P42858 1/20 0.47
GLA P06280 1/20 0.47
MAPK1 P28482 1/20 0.47
SLC18A3 Q16572 4/20 0.46
DRD2 P14416 1/20 0.46
MAPT P10636 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL8714788 0.95 CYP2C19 (0.47) CYP2C19CYP2D6OPRM1CYP1A2GAA
Fumaric Acid SCHEMBL8714787 0.95 CYP2C19 (0.47) CYP2C19CYP2D6OPRM1CYP1A2GAA
SCHEMBL8713866 0.93 OPRM1 (0.48) CYP2C19CYP2D6OPRM1CYP1A2GAA
SCHEMBL8714385 0.91 CYP2C19 (0.51) CYP2C19CYP2D6CYP1A2GAACYP2C9
Fumaric Acid SCHEMBL8711305 0.89 PTGIR (0.45) CYP2C19CYP2D6OPRM1CYP1A2GAA
Fumaric Acid SCHEMBL8711308 0.89 PTGIR (0.45) CYP2C19CYP2D6OPRM1CYP1A2GAA
SCHEMBL8712161 0.88 CYP2C9 (0.58) CYP2C19OPRM1CYP1A2GAACYP2C9
SCHEMBL8712582 0.88 OPRM1 (0.51) CYP2C19CYP2D6OPRM1CYP1A2GAA
SCHEMBL8711379 0.85 OPRM1 (0.48) CYP2C19CYP2D6OPRM1CYP1A2GAA
SCHEMBL8715758 0.84 HSD11B1 (0.48) CYP2C19CYP2D6CYP1A2GAACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5728835-A HYPOTENSIVE AGENTS; ANTIISCHEMIC AGENTS TOA EIYO, LTD. (JP) 1998-03-17 US disclosed
EP-0661266-A1 Substituted cyclic amine compounds as 5HT2 antagonists TOA EIYO LTD. (JP) 1995-07-05 EP disclosed