SCHEMBL8714804

SCHEMBL8714804

[CH]1CCCc2ccc(Cc3ccccc3)cc21

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.41
PARP11 Q9NR21 1/20 0.40
CALM1 P0DP23 1/20 0.40
PDK2 Q15119 1/20 0.37
TACR3 P29371 3/20 0.36
TACR1 P25103 2/20 0.36
HNF4A P41235 1/20 0.36
LTA4H P09960 4/20 0.35
NQO1 P15559 2/20 0.35
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5675962 0.78 PARP11 (0.50) IDH1PARP11CALM1TACR3TACR1
SCHEMBL2879790 0.77 NPC1 (0.39) PDK2TSHR
SCHEMBL27791814 0.77 PARP11 (0.49) IDH1PARP11CALM1TSHR
SCHEMBL5713934 0.75 CNR1 (0.38) PDK2
SCHEMBL5713702 0.73 GABRA1 (0.39) TSHR
SCHEMBL5713655 0.73 ESR1 (0.36)
SCHEMBL5714067 0.73 HRH3 (0.42) TSHR
SCHEMBL5714220 0.72 SKP2 (0.40)
SCHEMBL5713715 0.70 RELA (0.42) PDK2HNF4A
SCHEMBL19630481 0.69 TSHR (0.50) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5847006-A Therapeutic guanidines CAMBRIDGE NEUROSCIENCE, INC. (US) 1998-12-08 US disclosed
EP-0746316-A4 THERAPEUTIC GUANIDINES CAMBRIDGE NEUROSCIENCE INC (US) 1997-12-10 EP disclosed
EP-0746316-A1 THERAPEUTIC GUANIDINES CAMBRIDGE NEUROSCIENCE, INC. (US) 1996-12-11 EP disclosed
WO-1995014467-A1 THERAPEUTIC GUANIDINES CAMBRIDGE NEUROSCIENCE, INC. (US) 1995-06-01 WO disclosed