SCHEMBL8714982

SCHEMBL8714982

O=C1NC(=S)S/C1=C/Cc1cccc(Oc2ccccc2)c1

nearest known ligand 0.65

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 4/20 0.65
MMP3 P08254 3/20 0.65
ADAMTS5 Q9UNA0 10/20 0.56
GSK3B P49841 1/20 0.52
PTP4A3 O75365 1/20 0.49
AKR1B1 P15121 1/20 0.48
CA2 P00918 1/20 0.47
NAT1 P18440 1/20 0.47
EPHX1 P07099 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8311453 1.00 MMP13 (0.65) MMP13MMP3ADAMTS5GSK3BPTP4A3
SCHEMBL27479994 0.86 MEN1 (0.57) MMP13ADAMTS5GSK3BPTP4A3CA2
SCHEMBL18102998 0.84 NAT1 (0.59) MMP13MMP3ADAMTS5PTP4A3CA2
SCHEMBL8171894 0.84 NAT1 (0.59) MMP13MMP3ADAMTS5PTP4A3CA2
SCHEMBL8708384 0.80 PIM1 (0.61) MMP13MMP3ADAMTS5GSK3BPTP4A3
SCHEMBL8310456 0.80 PIM1 (0.61) MMP13MMP3ADAMTS5GSK3BPTP4A3
SCHEMBL8307763 0.80 NAT1 (0.61) MMP13MMP3ADAMTS5PTP4A3CA2
SCHEMBL8713697 0.80 NAT1 (0.61) MMP13MMP3ADAMTS5PTP4A3CA2
SCHEMBL8308267 0.79 MMP13 (1.00) MMP13MMP3ADAMTS5GSK3BAKR1B1
SCHEMBL1248886 0.79 MMP13 (1.00) MMP13MMP3ADAMTS5GSK3BAKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5716975-A NONTOXIC RHODANINE DERIVATIVES; ANTIDIABETIC AGENTS, CATHEPSIN D INHIBITORS, B-AMYLOID PROTEIN REDUCTION ELI LILLY AND COMPANY (US) 1998-02-10 US disclosed