Bromide

Bromide

SCHEMBL8715148

Br.NC1=Cc2cccc3cccc1c23

nearest known ligand 0.57

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.57
HSD17B10 Q99714 5/20 0.57
MAPT P10636 4/20 0.57
KDM4E B2RXH2 4/20 0.57
MEN1 O00255 3/20 0.57
KMT2A Q03164 3/20 0.57
HTT P42858 2/20 0.57
RXFP1 Q9HBX9 2/20 0.57
USP2 O75604 1/20 0.57
POLB P06746 1/20 0.57
ALOX15 P16050 1/20 0.57
MPI P34949 1/20 0.57
CACNA1B Q00975 1/20 0.57
APBA1 Q02410 1/20 0.57
MAPK1 P28482 4/20 0.50
CES2 O00748 1/20 0.43
BCHE P06276 1/20 0.43
CES1 P23141 1/20 0.43
MCL1 Q07820 1/20 0.43
TSHR P16473 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL131366 0.98 ALDH1A1 (0.59) ALDH1A1HSD17B10MAPTKDM4EMEN1
Hydrochloric Acid SCHEMBL8711400 0.96 ALDH1A1 (0.57) ALDH1A1HSD17B10MAPTKDM4EMEN1
SCHEMBL131080 0.75 MAPK1 (0.55) ALDH1A1HSD17B10MAPTKDM4EMEN1
SCHEMBL28962436 0.75 MAPK1 (0.55) ALDH1A1HSD17B10MAPTKDM4EMEN1
SCHEMBL8372344 0.72 ALDH1A1 (1.00) ALDH1A1HSD17B10MAPTKDM4EMEN1
SCHEMBL4073489 0.71 MAPK1 (0.74) ALDH1A1HSD17B10MAPTKDM4EMEN1
SCHEMBL131079 0.71 MAPK1 (0.52) ALDH1A1HSD17B10MAPTKDM4EMEN1
SCHEMBL130420 0.71 KMT2A (0.59) ALDH1A1HSD17B10MAPTKDM4EMEN1
SCHEMBL58539 0.71 MAPK1 (0.57) ALDH1A1HSD17B10MAPTKDM4EMEN1
SCHEMBL7557528 0.71 MAPK1 (0.52) ALDH1A1HSD17B10MAPTKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5847006-A Therapeutic guanidines CAMBRIDGE NEUROSCIENCE, INC. (US) 1998-12-08 US disclosed
EP-0746316-A4 THERAPEUTIC GUANIDINES CAMBRIDGE NEUROSCIENCE INC (US) 1997-12-10 EP disclosed
EP-0746316-A1 THERAPEUTIC GUANIDINES CAMBRIDGE NEUROSCIENCE, INC. (US) 1996-12-11 EP disclosed
WO-1995014467-A1 THERAPEUTIC GUANIDINES CAMBRIDGE NEUROSCIENCE, INC. (US) 1995-06-01 WO disclosed