SCHEMBL8715503

SCHEMBL8715503

COCOc1cc(F)c(Cl)cc1Br

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 7/20 0.36
HTR2B P41595 6/20 0.36
HTR2A P28223 6/20 0.36
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
ACLY P53396 1/20 0.32
MAPT P10636 1/20 0.32
SLC6A4 P31645 2/20 0.32
TAAR1 Q96RJ0 1/20 0.31
EGFR P00533 2/20 0.30
PIK3CD O00329 1/20 0.30
ABL1 P00519 1/20 0.30
HCK P08631 1/20 0.30
SRC P12931 1/20 0.30
KDR P35968 1/20 0.30
PIK3CA P42336 1/20 0.30
PIK3CB P42338 1/20 0.30
MTOR P42345 1/20 0.30
PIK3CG P48736 1/20 0.30
EPHB4 P54760 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29447054 0.93 HTR2A (0.33) HTR2CHTR2BHTR2AKDM4EALDH1A1
SCHEMBL4520961 0.93 HTR2A (0.33) HTR2CHTR2BHTR2AKDM4EALDH1A1
SCHEMBL26932098 0.81 HTR2A (0.42) HTR2CHTR2AKDM4EALDH1A1MAPT
SCHEMBL18768219 0.81 HTR2A (0.37) HTR2CHTR2BHTR2AALDH1A1MAPT
SCHEMBL31167218 0.80 ALDH1A1 (0.34) HTR2CHTR2AKDM4EALDH1A1MAPT
SCHEMBL4148256 0.80 HTR2A (0.44) HTR2CHTR2BHTR2ATAAR1PRKDC
SCHEMBL31566995 0.80 HTR2A (0.44) HTR2CHTR2BHTR2ATAAR1PRKDC
SCHEMBL29283664 0.79 ACLY (0.37) HTR2CHTR2AKDM4EALDH1A1ACLY
SCHEMBL15980355 0.79 HTR2A (0.39) HTR2CHTR2AKDM4EALDH1A1MAPT
SCHEMBL18751319 0.77 HTR2A (0.35) HTR2CHTR2BHTR2ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5716971-A FOR TREATMENT OF ANGINA PECTORIS AND HYPERTENSION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-10 US disclosed
EP-0623597-B1 Pyridine derivatives, with potassium channel opening activity TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-10-22 EP disclosed
EP-0623597-A1 Pyridine derivatives, with potassium channel opening activity Takeda Chemical Industries, Ltd. (JP) 1994-11-09 EP disclosed