SCHEMBL8716491

SCHEMBL8716491

CC(=O)Oc1cccnc1/C(=N\OC(C)(C)C)c1cc(C(F)(F)F)ccc1O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.41
USP2 O75604 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
CYP2C19 P33261 1/20 0.41
HSD17B10 Q99714 1/20 0.41
BACE1 P56817 1/20 0.37
TLR7 Q9NYK1 3/20 0.36
SCN8A Q9UQD0 2/20 0.35
SCN10A Q9Y5Y9 2/20 0.35
TBXA2R P21731 2/20 0.33
CNR2 P34972 1/20 0.33
LRRK2 Q5S007 1/20 0.33
SRPK3 Q9UPE1 1/20 0.33
P2RY1 P47900 1/20 0.32
COMT P21964 1/20 0.32
RXRA P19793 2/20 0.32
NR1H2 P55055 2/20 0.32
NR1H3 Q13133 2/20 0.32
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8716493 1.00 KDM4E (0.41) KDM4EUSP2ALDH1A1HPGDCYP2C19
SCHEMBL8709612 0.85 TLR7 (0.42) KDM4EALDH1A1TLR7SCN8ASCN10A
SCHEMBL8709608 0.85 TLR7 (0.42) KDM4EALDH1A1TLR7SCN8ASCN10A
SCHEMBL8713451 0.80 ELANE (0.34) KDM4ECYP2C19TLR7TBXA2RCNR2
SCHEMBL8713450 0.80 ELANE (0.34) KDM4ECYP2C19TLR7TBXA2RCNR2
SCHEMBL8709311 0.74 ALDH1A1 (0.34) KDM4EALDH1A1TLR7MAPTHTT
SCHEMBL8709309 0.74 ALDH1A1 (0.34) KDM4EALDH1A1TLR7MAPTHTT
SCHEMBL8709643 0.72 MEN1 (0.35) KDM4EALDH1A1HPGDCYP2C19TLR7
SCHEMBL8714961 0.71 TLR7 (0.36) KDM4ECYP2C19TLR7RXRA
SCHEMBL8714957 0.71 TLR7 (0.36) KDM4ECYP2C19TLR7RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5716971-A FOR TREATMENT OF ANGINA PECTORIS AND HYPERTENSION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-10 US disclosed
EP-0623597-B1 Pyridine derivatives, with potassium channel opening activity TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-10-22 EP disclosed
EP-0623597-A1 Pyridine derivatives, with potassium channel opening activity Takeda Chemical Industries, Ltd. (JP) 1994-11-09 EP disclosed