SCHEMBL8718599

SCHEMBL8718599

O[C@@H](C[C@@H]1CO1)c1ccc(F)cc1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
PDE2A O00408 2/20 0.36
SLC6A2 P23975 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2D6 P10635 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
HSD11B1 P28845 1/20 0.33
MC4R P32245 1/20 0.33
IDO1 P14902 1/20 0.33
TDO2 P48775 1/20 0.33
IDH1 O75874 1/20 0.32
GRIN2B Q13224 1/20 0.32
ADRB2 P07550 1/20 0.32
HSD17B10 Q99714 1/20 0.32
ADRA2A P08913 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9721750 0.76 KDM4E (0.46) HTR2AHTR2CIDO1
SCHEMBL12303658 0.73 CES2 (0.49) CES2CES1PDE2ASLC6A2CYP3A4
SCHEMBL5225559 0.73 ADRA2C (0.57) CES2CES1PDE2ASLC6A2CYP3A4
SCHEMBL7145782 0.73 ADRA2C (0.57) CES2CES1PDE2ASLC6A2CYP3A4
SCHEMBL17121793 0.72 CES2 (0.39) CES2CES1CYP3A4ADRB2HSD17B10
SCHEMBL10306200 0.72 CES2 (0.47) CES2CES1PDE2ASLC6A2CYP3A4
SCHEMBL14539581 0.72 CES2 (0.47) CES2CES1PDE2ASLC6A2CYP3A4
SCHEMBL28155953 0.72 CES2 (0.47) CES2CES1PDE2ASLC6A2CYP3A4
Hydrochloric Acid SCHEMBL5354434 0.72 KDM4E (0.58) CES2CES1PDE2ASLC6A2CYP3A4
SCHEMBL8580203 0.71 CES2 (0.41) CES2CES1SLC6A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0567982-B1 Azole compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1998-07-01 EP disclosed
US-5466820-A Fungicides TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-11-14 US disclosed
US-5371101-A Fungicides TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-12-06 US disclosed
EP-0567982-A1 Azole compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1993-11-03 EP disclosed