SCHEMBL8719491

SCHEMBL8719491

CCCCCCCCCCCCCCCCCCN(CCCCCCCCCCCCCCCCCC)C(=O)CN(CCN(CC(=O)OC(C)(C)C)CC(=O)OC(C)(C)C)CCN(CC(=O)OC(C)(C)C)CC(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 8/20 0.40
CA1 P00915 8/20 0.40
CA2 P00918 6/20 0.40
CA4 P22748 2/20 0.40
DNM1 Q05193 1/20 0.35
CA9 Q16790 3/20 0.34
CA14 Q9ULX7 1/20 0.33
NAAA Q02083 1/20 0.33
DGKA P23743 1/20 0.33
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33
KDM5A P29375 3/20 0.33
RAD52 P43351 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
PHF8 Q9UPP1 2/20 0.32
ZDHHC20 Q5W0Z9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10181438 0.84 CA12 (0.48) CA12CA1CA2CA4DNM1
SCHEMBL22667659 0.84 CA12 (0.48) CA12CA1CA2CA4DNM1
SCHEMBL16558064 0.83 DNM1 (0.39) CA12CA1DNM1CA14NAAA
SCHEMBL7567930 0.83 CA12 (0.37) CA12CA1DNM1CA9CA14
SCHEMBL15197286 0.82 CA12 (0.38) CA12CA1CA2CA4CA9
SCHEMBL22506543 0.79 DNM1 (0.36) CA12CA1DNM1CA14NAAA
SCHEMBL4061196 0.79 CA12 (0.52) CA12CA1CA2CA4DNM1
SCHEMBL19458 0.79 TDP1 (0.42) CA12CA1CA2CA4CA14
SCHEMBL21838011 0.79 CA14 (0.46) CA12CA1CA2DNM1CA9
SCHEMBL19040823 0.79 DNM1 (0.50) DNM1DGKAKDM5APHF8KDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5730956-A DTPA di-alkyl monoamides for x-ray and MRI SCHERING AKTIENGESELLSCHAFT (DE) 1998-03-24 US disclosed
EP-0810990-A1 SUBSTITUTED DTPA MONOAMIDES OF CENTRAL CARBOXYLIC ACIDS AND METAL COMPLEXES THEREOF, PHARMACEUTICALS CONTAINING THESE COMPLEXES, DIAGNOSTIC AND THERAPEUTIC USES THEREOF AND METHODS FOR PREPARING THE COMPLEXES AND PHARMACEUTICALS SCHERING AKTIENGESELLSCHAFT (DE) 1997-12-10 EP disclosed
US-5679852-A Process for the production of DTPA-monoamides of the central carboxylic acid and their use as pharmaceutical agents SCHERING AKTIENGESELLSCHAFT (DE) 1997-10-21 US disclosed
US-5676923-A SOLUBLE, STABLE, ORGAN-SPECIFIC NUCLEAR MAGNETIC RESONANCE CONTRAST AGENT SCHERING AKTIENGESELLSCHAFT (DE) 1997-10-14 US disclosed
WO-1996026182-A1 SUBSTITUTED DTPA MONOAMIDES OF CENTRAL CARBOXYLIC ACIDS AND METAL COMPLEXES THEREOF, PHARMACEUTICALS CONTAINING THESE COMPLEXES, DIAGNOSTIC AND THERAPEUTIC USES THEREOF AND METHODS FOR PREPARING THE COMPLEXES AND PHARMACEUTICALS SCHERING AKTIENGESELLSCHAFT (DE) 1996-08-29 WO disclosed