SCHEMBL8723573

SCHEMBL8723573

[CH]c1c(Cl)c(Cl)cc2ccccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 5/20 0.45
CYP1A2 P05177 3/20 0.43
ALDH1A1 P00352 3/20 0.40
HSD17B10 Q99714 2/20 0.39
HIF1A Q16665 1/20 0.39
CYP1B1 Q16678 1/20 0.39
L3MBTL1 Q9Y468 3/20 0.39
CCR1 P32246 1/20 0.37
CCR8 P51685 1/20 0.37
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
AHR P35869 1/20 0.36
TRPM4 Q8TD43 1/20 0.35
TSHR P16473 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
HTR2A P28223 1/20 0.34
NQO2 P16083 1/20 0.34
MAPT P10636 1/20 0.34
APAF1 O14727 1/20 0.34
TDP2 O95551 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8723579 1.00 CYP2A6 (0.45) CYP2A6CYP1A2ALDH1A1HSD17B10HIF1A
SCHEMBL29629107 0.79 CYP2A6 (0.56) CYP2A6CYP1A2ALDH1A1HSD17B10HIF1A
SCHEMBL1039782 0.79 CYP2A6 (0.56) CYP2A6CYP1A2ALDH1A1HSD17B10HIF1A
SCHEMBL1673423 0.76 ALDH1A1 (0.50) CYP2A6CYP1A2ALDH1A1HSD17B10HIF1A
SCHEMBL30499577 0.74 HSD17B10 (0.48) CYP2A6CYP1A2ALDH1A1HSD17B10HIF1A
SCHEMBL27002361 0.74 CYP2A6 (0.50) CYP2A6CYP1A2ALDH1A1HSD17B10HIF1A
SCHEMBL29244212 0.74 CYP2A6 (0.45) CYP2A6CYP1A2ALDH1A1HSD17B10HIF1A
SCHEMBL10877466 0.74 CYP2A6 (0.45) CYP2A6CYP1A2ALDH1A1HSD17B10HIF1A
SCHEMBL554286 0.74 HSD17B10 (0.48) CYP2A6CYP1A2ALDH1A1HSD17B10HIF1A
SCHEMBL5610395 0.74 CYP2A6 (0.45) CYP2A6CYP1A2ALDH1A1HSD17B10HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0609058-B1 Hexahydronaphthalene ester derivatives, their preparation and their therapeutic uses SANKYO CO (JP) 1998-12-09 EP disclosed
US-5491167-A INHIBITORS OF CHOLESTEROL BIOSYNTHESIS SANKYO COMPANY, LIMITED (JP) 1996-02-13 US disclosed
EP-0609058-A2 Hexahydronaphthalene ester derivatives, their preparation and their therapeutic uses SANKYO COMPANY LIMITED (JP) 1994-08-03 EP disclosed