SCHEMBL872527

SCHEMBL872527

O=C(O)NCCOc1ccsc1C(=O)Nc1ncc([N+](=O)[O-])s1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.52
RAB9A P51151 7/20 0.52
MEN1 O00255 5/20 0.52
KMT2A Q03164 5/20 0.52
PKM P14618 5/20 0.52
ATG4B Q9Y4P1 7/20 0.51
STAT3 P40763 7/20 0.48
ALDH1A1 P00352 2/20 0.47
MAPT P10636 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
CDK2 P24941 2/20 0.47
GSK3A P49840 2/20 0.47
GSK3B P49841 2/20 0.47
DYRK1A Q13627 1/20 0.47
HIPK4 Q8NE63 1/20 0.47
CLK4 Q9HAZ1 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
MLNR O43193 1/20 0.47
NR1I2 O75469 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10211140 0.89 RAB9A (0.53) NPC1RAB9AMEN1KMT2APKM
SCHEMBL375797 0.87 NPC1 (0.47) NPC1RAB9AMEN1KMT2APKM
Hydrochloric Acid SCHEMBL375506 0.86 NPC1 (0.55) NPC1RAB9AMEN1KMT2APKM
SCHEMBL876378 0.76 STAT3 (0.64) NPC1RAB9AMEN1KMT2APKM
SCHEMBL10257101 0.74 NPC1 (0.49) NPC1RAB9AMEN1KMT2APKM
SCHEMBL10211139 0.71 STAT3 (0.67) NPC1RAB9AMEN1KMT2APKM
SCHEMBL29056983 0.71 STAT3 (0.53) NPC1RAB9AMEN1KMT2APKM
SCHEMBL376276 0.71 MEN1 (0.62) NPC1RAB9AMEN1KMT2APKM
SCHEMBL30142671 0.70 STAT3 (0.66) NPC1RAB9AMEN1KMT2APKM
SCHEMBL1804666 0.69 NPC1 (0.76) NPC1RAB9AMEN1KMT2APKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2632460-A2 COMPOSITIONS AND METHODS FOR TREATING TUBERCULOSIS University Of Virginia Patent Foundation (US) 2013-09-04 EP disclosed
WO-2012040170-A2 COMPOSITIONS AND METHODS FOR TREATING TUBERCULOSIS UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2012-03-29 WO disclosed