SCHEMBL8725283

SCHEMBL8725283

CC(c1ccc(Nc2cc[c]cc2)cc1)N1CCCC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.42
LTA4H P09960 1/20 0.38
MC4R P32245 1/20 0.38
CYP26A1 O43174 1/20 0.37
CHRM2 P08172 7/20 0.36
CHRM1 P11229 7/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
CYP3A4 P08684 2/20 0.34
CYP2C9 P11712 1/20 0.34
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
MBTD1 Q05BQ5 1/20 0.34
L3MBTL3 Q96JM7 1/20 0.34
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
THRB P10828 1/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33
ALOX12 P18054 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3030261 0.84 CYP2D6 (0.52) CYP2D6LTA4HMC4RCHRM2CHRM1
SCHEMBL6233324 0.83 CYP2D6 (0.50) CYP2D6LTA4HMC4RCHRM2CHRM1
SCHEMBL8725280 0.81 CYP2D6 (0.44) CYP2D6LTA4HMC4RCYP26A1CHRM2
SCHEMBL16982012 0.73 CYP2D6 (0.56) CYP2D6LTA4HMC4RCHRM2CHRM1
SCHEMBL16270668 0.71 CHRM2 (0.54) CYP2D6LTA4HMC4RCHRM2CHRM1
SCHEMBL2735673 0.71 CHRM2 (0.54) CYP2D6LTA4HMC4RCHRM2CHRM1
SCHEMBL12781671 0.70 CHRM2 (0.57) CYP2D6LTA4HMC4RCHRM2CHRM1
SCHEMBL2236588 0.70 NCF1 (0.54) CYP2D6LTA4HMC4RCHRM2CHRM1
SCHEMBL3041069 0.70 CYP2D6 (0.52) CYP2D6LTA4HMC4RCHRM2CHRM1
SCHEMBL6872559 0.70 CYP2D6 (0.52) CYP2D6LTA4HMC4RCHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832091-A1 C-4' MODIFIED ADENOSINE KINASE INHIBITORS GENSIA, INC. (US) 1998-04-01 EP disclosed
WO-1996040705-A1 C-4' MODIFIED ADENOSINE KINASE INHIBITORS GENSIA SICOR (US) 1996-12-19 WO disclosed