SCHEMBL8725280

SCHEMBL8725280

CC(c1ccc(Nc2[c]cccc2)cc1)N1CCCC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.44
LTA4H P09960 1/20 0.40
MC4R P32245 1/20 0.40
CHRM2 P08172 6/20 0.38
CHRM1 P11229 6/20 0.38
CYP26A1 O43174 1/20 0.36
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35
OPRL1 P41146 1/20 0.35
CYP3A4 P08684 4/20 0.33
CYP1A2 P05177 3/20 0.33
CYP2C9 P11712 3/20 0.33
KCNA5 P22460 3/20 0.33
CYP2C19 P33261 3/20 0.33
KCNH2 Q12809 3/20 0.33
MBTD1 Q05BQ5 1/20 0.33
L3MBTL3 Q96JM7 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8725283 0.81 CYP2D6 (0.42) CYP2D6LTA4HMC4RCHRM2CHRM1
SCHEMBL8722503 0.79 NFKB1 (0.42) CYP3A4ALDH1A1LMNATHRBALOX15
SCHEMBL7795568 0.72 KCNA5 (0.37) CYP2D6CYP3A4CYP1A2CYP2C9KCNA5
SCHEMBL3030261 0.71 CYP2D6 (0.52) CYP2D6LTA4HMC4RCHRM2CHRM1
SCHEMBL8983627 0.71 CYP2D6 (0.83) CYP2D6LTA4HMC4RCHRM2CHRM1
SCHEMBL8983562 0.71 CYP2D6 (0.83) CYP2D6LTA4HMC4RCHRM2CHRM1
SCHEMBL7097730 0.71 CYP2D6 (0.83) CYP2D6LTA4HMC4RCHRM2CHRM1
SCHEMBL2587778 0.71 CYP2D6 (0.42) CYP2D6LTA4HMC4RCHRM2CHRM1
SCHEMBL6233324 0.70 CYP2D6 (0.50) CYP2D6LTA4HMC4RCHRM2CHRM1
SCHEMBL6418064 0.70 HPGD (0.54) ALDH1A1LMNAALOX15TSHRALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832091-A1 C-4' MODIFIED ADENOSINE KINASE INHIBITORS GENSIA, INC. (US) 1998-04-01 EP disclosed
WO-1996040705-A1 C-4' MODIFIED ADENOSINE KINASE INHIBITORS GENSIA SICOR (US) 1996-12-19 WO disclosed