SCHEMBL8725874

SCHEMBL8725874

N#CC(C(=O)NN)c1ccccn1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.57
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
GAA P10253 2/20 0.57
ALDH1A1 P00352 6/20 0.45
CTSD P07339 1/20 0.42
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.38
P2RX7 Q99572 1/20 0.37
KDM4E B2RXH2 5/20 0.36
LMNA P02545 2/20 0.36
OPRK1 P41145 2/20 0.36
HTT P42858 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
SLC6A3 Q01959 2/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
S1PR1 P21453 1/20 0.35
S1PR3 Q99500 1/20 0.35
ABCB11 O95342 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL783597 0.80 KMT2A (0.63) SMN1; SMN2MEN1KMT2AGAAALDH1A1
SCHEMBL19668743 0.79 SMN1; SMN2 (0.66) SMN1; SMN2MEN1KMT2AGAAALDH1A1
SCHEMBL4361229 0.79 SMN1; SMN2 (0.66) SMN1; SMN2MEN1KMT2AGAAALDH1A1
SCHEMBL31724491 0.78 KMT2A (0.74) SMN1; SMN2MEN1KMT2AGAAALDH1A1
SCHEMBL15745601 0.76 CYP1A2 (0.55) SMN1; SMN2MEN1KMT2AGAAALDH1A1
SCHEMBL11689283 0.76 CTSD (0.42) SMN1; SMN2MEN1KMT2AGAAALDH1A1
SCHEMBL21378747 0.76 CYP1A2 (0.55) SMN1; SMN2MEN1KMT2AGAAALDH1A1
SCHEMBL21378793 0.76 CYP1A2 (0.55) SMN1; SMN2MEN1KMT2AGAAALDH1A1
SCHEMBL9574957 0.75 CTSD (0.63) SMN1; SMN2MEN1KMT2AGAAALDH1A1
SCHEMBL13516453 0.73 SMN1; SMN2 (1.00) SMN1; SMN2MEN1KMT2AGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0876370-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-11-11 EP disclosed
WO-1997025325-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-07-17 WO disclosed