SCHEMBL8726328

SCHEMBL8726328

C[C@@]12CCC[C@H]1[C@@H]1CCN3CC(=O)CC[C@]3(C)[C@@H]1CC2

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 4/20 0.43
MBOAT4 Q96T53 3/20 0.39
CDK5 Q00535 1/20 0.39
CDK5R1 Q15078 1/20 0.39
NR1I3 Q14994 1/20 0.36
SRD5A2 P31213 2/20 0.34
GRIN1 Q05586 4/20 0.34
GRIN2B Q13224 4/20 0.34
SHBG P04278 1/20 0.33
STS P08842 1/20 0.31
AKR1B10 O60218 1/20 0.30
AKR1B1 P15121 1/20 0.30
OR51E2 Q9H255 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9546874 0.71 AR (0.34) CYP19A1SRD5A2SHBG
SCHEMBL27248784 0.68 AKR1B10 (0.65) CYP19A1MBOAT4CDK5CDK5R1NR1I3
SCHEMBL9541973 0.68 AKR1B10 (0.65) CYP19A1MBOAT4CDK5CDK5R1NR1I3
SCHEMBL27607786 0.68 AKR1B10 (0.65) CYP19A1MBOAT4CDK5CDK5R1NR1I3
SCHEMBL19877200 0.68 AKR1B10 (0.65) CYP19A1MBOAT4CDK5CDK5R1NR1I3
SCHEMBL24151978 0.68 AKR1B10 (0.65) CYP19A1MBOAT4CDK5CDK5R1NR1I3
SCHEMBL4572602 0.68 AKR1B10 (0.65) CYP19A1MBOAT4CDK5CDK5R1NR1I3
SCHEMBL1962644 0.68 AKR1B10 (0.65) CYP19A1MBOAT4CDK5CDK5R1NR1I3
SCHEMBL1651202 0.68 AKR1B10 (0.65) CYP19A1MBOAT4CDK5CDK5R1NR1I3
SCHEMBL1427282 0.68 AKR1B10 (0.65) CYP19A1MBOAT4CDK5CDK5R1NR1I3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5710275-A ENZYME AND HORMONE INHIBITORS MERCK & CO., INC. (US) 1998-01-20 US disclosed
EP-0649431-A4 17-AMINO SUBSTITUTED 4-AZASTEROID 5-G(A)-REDUCTASE INHIBITORS. 1995-05-03 EP disclosed
EP-0649431-A1 17-AMINO SUBSTITUTED 4-AZASTEROID 5$g(a)-REDUCTASE INHIBITORS MERCK & CO. INC. (US) 1995-04-26 EP disclosed
WO-1993023038-A1 17-AMINO SUBSTITUTED 4-AZASTEROID 5α-REDUCTASE INHIBITORS MERCK & CO., INC. (US) 1993-11-25 WO disclosed