SCHEMBL8727017

SCHEMBL8727017

Cn1c(CC(=O)O)ccc1C(=O)Cc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 3/20 0.54
AKR1B1 P15121 2/20 0.54
PTGS2 P35354 2/20 0.54
CXCL8 P10145 1/20 0.54
GLO1 Q04760 1/20 0.54
HDAC3 O15379 1/20 0.52
HDAC4 P56524 1/20 0.52
HDAC1 Q13547 1/20 0.52
HDAC7 Q8WUI4 1/20 0.52
HDAC2 Q92769 1/20 0.52
HDAC8 Q9BY41 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
HDAC9 Q9UKV0 1/20 0.52
HDAC5 Q9UQL6 1/20 0.52
KDM4E B2RXH2 2/20 0.49
L3MBTL1 Q9Y468 2/20 0.49
LMNA P02545 2/20 0.43
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
ABCC4 O15439 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8732219 0.91 PTGS1 (0.56) PTGS1AKR1B1PTGS2CXCL8GLO1
SCHEMBL8732105 0.86 AKR1B1 (0.50) PTGS1AKR1B1PTGS2CXCL8GLO1
SCHEMBL17486795 0.85 HDAC3 (0.48) PTGS1AKR1B1PTGS2CXCL8GLO1
SCHEMBL8732035 0.84 HDAC1 (0.50) PTGS1AKR1B1PTGS2CXCL8GLO1
SCHEMBL8732100 0.83 MAPT (0.50) PTGS1AKR1B1PTGS2CXCL8GLO1
SCHEMBL10940661 0.81 HDAC8 (0.56) AKR1B1HDAC3HDAC4HDAC1HDAC7
SCHEMBL2237360 0.79 PTGS2 (0.77) PTGS1AKR1B1PTGS2CXCL8GLO1
SCHEMBL8731019 0.78 PTGS2 (0.70) PTGS1AKR1B1PTGS2CXCL8GLO1
SCHEMBL8729681 0.78 PTGS2 (0.70) PTGS1AKR1B1PTGS2CXCL8GLO1
SCHEMBL2237110 0.78 PTGS2 (0.61) PTGS1AKR1B1PTGS2CXCL8GLO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0783488-A4 FIVE MEMBERED HETEROCYCLIC COMPOUNDS ONO PHARMACEUTICAL CO (JP) 1998-01-07 EP claimed
EP-0783488-A1 FIVE MEMBERED HETEROCYCLIC COMPOUNDS ONO PHARMACEUTICAL CO., LTD. (JP) 1997-07-16 EP claimed
WO-1996010013-A1 FIVE MEMBERED HETEROCYCLIC COMPOUNDS ONO PHARMACEUTICAL CO., LTD. (JP) 1996-04-04 WO claimed