SCHEMBL8728129

SCHEMBL8728129

CCCC(C)CC(N=C=O)C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 1/20 0.38
AKR1A1 P14550 1/20 0.38
CHRM3 P20309 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
ADRA1A P35348 1/20 0.38
HRH1 P35367 1/20 0.38
DRD3 P35462 1/20 0.38
SLC6A3 Q01959 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
TSHR P16473 1/20 0.34
GRIK1 P39086 1/20 0.34
SLC1A3 P43003 1/20 0.34
SLC1A2 P43004 1/20 0.34
SLC1A1 P43005 1/20 0.34
GRIK2 Q13002 1/20 0.34
ACE2 Q9BYF1 1/20 0.33
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6101629 0.83 CHRM1 (0.44) CHRM1AKR1A1CHRM3HTR2AHTR2C
SCHEMBL7701831 0.79 RNPEP (0.41) ADRA1ASLC1A3SLC1A2MAPT
SCHEMBL6056700 0.79 RNPEP (0.41) ADRA1ASLC1A3SLC1A2MAPT
SCHEMBL11158578 0.78 CYP3A4 (0.31) TSHRMAPT
Water SCHEMBL27284531 0.77 RNPEP (0.40) ADRA1ASLC1A3SLC1A2MAPT
SCHEMBL28822953 0.77 RNPEP (0.31)
SCHEMBL4906428 0.76 CA2 (0.45) CHRM1AKR1A1CHRM3HTR2AHTR2C
SCHEMBL592033 0.76 CA2 (0.45) CHRM1AKR1A1CHRM3HTR2AHTR2C
SCHEMBL4789164 0.75 ALDH1A1 (0.33) ACE2
SCHEMBL10746086 0.75 TSHR (0.36) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0816309-A1 Scavenger assisted combinatorial process for preparing libraries of urea and thiourea compounds ELI LILLY AND COMPANY (US) 1998-01-07 EP disclosed