SCHEMBL8728352

SCHEMBL8728352

CC(=O)Oc1ccc2c(CBr)cc(=O)oc2c1.COc1cc2oc(=O)cc(CBr)c2cc1OC

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.57
ALDH1A1 P00352 7/20 0.57
GAA P10253 6/20 0.57
GLA P06280 5/20 0.57
LCK P06239 1/20 0.54
HPGD P15428 3/20 0.53
POLB P06746 2/20 0.51
CA12 O43570 2/20 0.51
CA9 Q16790 2/20 0.51
TDP1 Q9NUW8 1/20 0.51
CYP2D6 P10635 2/20 0.50
KMT2A Q03164 3/20 0.48
CASP1 P29466 3/20 0.47
CASP7 P55210 3/20 0.47
HSD17B10 Q99714 3/20 0.47
MAPT P10636 3/20 0.47
HSP90AA1 P07900 1/20 0.47
HSP90AB1 P08238 1/20 0.47
ALPG P10696 1/20 0.47
ALOX15 P16050 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL68231 0.91 KDM4E (0.68) KDM4EALDH1A1GAAGLALCK
SCHEMBL31344274 0.84 MCL1 (0.47) KDM4EALDH1A1GLALCKHPGD
SCHEMBL67273 0.84 MCL1 (0.47) KDM4EALDH1A1GLALCKHPGD
SCHEMBL8654964 0.83 KDM4E (0.56) KDM4EALDH1A1GAAGLALCK
SCHEMBL29443248 0.81 CYP2D6 (0.72) KDM4EALDH1A1LCKHPGDPOLB
SCHEMBL67779 0.81 CYP2D6 (0.72) KDM4EALDH1A1LCKHPGDPOLB
SCHEMBL8863327 0.81 KDM4E (0.65) KDM4EALDH1A1GAAGLALCK
SCHEMBL6996933 0.80 KDM4E (0.57) KDM4EALDH1A1GAAGLALCK
Phosphine SCHEMBL17375055 0.80 CYP2D6 (0.70) KDM4EALDH1A1LCKHPGDPOLB
SCHEMBL8675851 0.78 KDM4E (0.53) KDM4EALDH1A1GAAGLALCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998008839-A1 COMBINATORIAL PROCESS FOR PREPARING SUBSTITUTED THIOPHENE LIBRARIES ELI LILLY AND COMPANY (US) 1998-03-05 WO disclosed