SCHEMBL8728401

SCHEMBL8728401

NCCc1ccc(OCP(=O)(O)C2CCCCC2)cc1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.39
NUDT1 P36639 1/20 0.39
BACE1 P56817 1/20 0.39
PTPN1 P18031 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
TPSAB1 Q15661 1/20 0.38
TPSD1 Q9BZJ3 1/20 0.38
TPSG1 Q9NRR2 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8729727 0.85 S1PR4 (0.43) MEN1KMT2A
SCHEMBL8727043 0.81 SLC6A4 (0.43) PTPN1TAAR1
SCHEMBL8584969 0.80 CYP2C9 (0.56) MEN1KMT2A
SCHEMBL8732769 0.78 PTPN1 (0.60) MAOBPTPN1TAAR1
SCHEMBL8729734 0.77 MEN1 (0.38) MAOBNUDT1BACE1TAAR1MEN1
SCHEMBL8729155 0.76 NAMPT (0.43) PTPN1MEN1KMT2A
SCHEMBL8730020 0.74 MEN1 (0.40) TAAR1MEN1KMT2A
SCHEMBL8728408 0.74 TAAR1 (0.42) MAOBNUDT1BACE1TAAR1
SCHEMBL8758157 0.74 KMT2A (0.47) MEN1KMT2A
SCHEMBL5449632 0.74 ADRB3 (0.65)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5726165-A HYPOGLYCEMIC AGENTS; DIETETICS; GASTROINTESTINAL DISORDERS SMITHKLINE BEECHAM P.L.C. (GB) 1998-03-10 US disclosed
EP-0772585-A1 ARYLOXY AND ARYLTHIOPROPANOLAMINE DERIVATIVES USEFUL AS BETA 3-ADRENORECEPTOR AGONISTS AND ANTAGONISTS OF THE BETA 1 AND BETA 2-ADRENORECEPTORS AND PHARMACEUTICAL COMPOSITION THEREOF SMITHKLINE BEECHAM PLC (GB) 1997-05-14 EP disclosed
WO-1996004233-A1 ARYLOXY AND ARYLTHIOPROPANOLAMINE DERIVATIVES USEFUL AS BETA 3-ADRENORECEPTOR AGONISTS AND ANTAGONISTS OF THE BETA 1 AND BETA 2-ADRENORECEPTORS AND PHARMACEUTICAL COMPOSITION THEREOF SMITHKLINE BEECHAM PLC (GB) 1996-02-15 WO disclosed