SCHEMBL8729433

SCHEMBL8729433

CN(C(=O)NC(CC(N)=O)C(=O)NC(Cc1ccccc1)C(O)CNCCc1ccccc1)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BCHE P06276 5/20 0.43
BACE1 P56817 11/20 0.43
SLC6A11 P48066 1/20 0.43
CTSD P07339 2/20 0.41
BACE2 Q9Y5Z0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8735254 0.92 BACE1 (0.53) BCHEBACE1SLC6A11CTSD
SCHEMBL8734441 0.91 CTSD (0.44) BCHEBACE1SLC6A11CTSD
SCHEMBL8735226 0.91 BACE1 (0.44) BCHEBACE1SLC6A11CTSD
SCHEMBL8732160 0.90 BACE1 (0.46) BCHEBACE1SLC6A11
SCHEMBL8732197 0.88 BCHE (0.59) BCHEBACE1SLC6A11
SCHEMBL8732007 0.87 BACE1 (0.49) BCHEBACE1SLC6A11CTSDBACE2
SCHEMBL8729328 0.85 BACE1 (0.50) BCHEBACE1SLC6A11CTSD
SCHEMBL9050282 0.83 ADORA3 (0.42) BCHEBACE1
SCHEMBL8984684 0.83 ADORA3 (0.42) BCHEBACE1CTSD
SCHEMBL8840191 0.80 PSEN1 (0.43) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5708004-A ENZYME INHIBITORS FOR TREATMENT OF AIDS MONSANTO COMPANY (US) 1998-01-13 US disclosed
US-5703076-A TREATING HIV, AIDS G. D. SEARLE & CO. (US) 1997-12-30 US disclosed
US-5698569-A Retroviral protease inhibitors G. D. SEARLE & CO. (US) 1997-12-16 US disclosed
US-5510349-A HUMAN IMMUNODEFICIENCY VIRUS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5510487-A TREATING HUMAN IMMUNODEFICIENCY VIRUS INFECTIONS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5510378-A Retroviral protease inhibitors G.D. SEARLE & CO. (US) 1996-04-23 US disclosed