SCHEMBL873112

SCHEMBL873112

C[C@]1(O)C(n2cc(Br)c3c(N)ncnc32)O[C@H](CO)[C@H]1O

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.65
ADK P55263 7/20 0.56
ADORA3 P0DMS8 4/20 0.47
ADORA2B P29275 2/20 0.47
ADORA1 P30542 2/20 0.47
METTL3 Q86U44 5/20 0.47
ADA P00813 1/20 0.45
DOT1L Q8TEK3 1/20 0.44
NPC1 O15118 1/20 0.44
GALR3 O60755 1/20 0.44
S1PR4 O95977 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
S1PR1 P21453 1/20 0.44
HTT P42858 1/20 0.44
RAB9A P51151 1/20 0.44
PAX8 Q06710 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL474780 1.00 ADORA2A (0.65) ADORA2AADKADORA3ADORA2BADORA1
SCHEMBL2788245 0.89 ADK (0.56) ADORA2AADKMETTL3DOT1LNPC1
SCHEMBL2788742 0.89 ADK (0.56) ADORA2AADKMETTL3DOT1LNPC1
SCHEMBL3229703 0.89 ADORA2A (0.67) ADORA2AADKADORA3ADORA2BADORA1
SCHEMBL474796 0.88 ADORA2A (0.66) ADORA2AADKADORA3ADORA2BADORA1
SCHEMBL873435 0.88 ADORA2A (0.66) ADORA2AADKADORA3ADORA2BADORA1
SCHEMBL18200214 0.88 ADORA2A (0.66) ADORA2AADKADORA3ADORA2BADORA1
SCHEMBL14544819 0.88 ADORA2A (0.66) ADORA2AADKADORA3ADORA2BADORA1
SCHEMBL15241391 0.88 ADORA2A (0.66) ADORA2AADKADORA3ADORA2BADORA1
SCHEMBL24837545 0.87 ADORA2A (0.65) ADORA2AADKADORA3ADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2618665-A1 HCV NS3 PROTEASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2013-07-31 EP disclosed
EP-1476169-B1 Inhibiting orthopoxvirus replication with nucleoside compounds MERCK SHARP & DOHME (US) 2013-03-20 EP disclosed
WO-2012040040-A1 HCV NS3 PROTEASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-03-29 WO disclosed