SCHEMBL873200

SCHEMBL873200

O=C(Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3CCCN3C(=O)C3=CC3)cc2)cc1)[C@@H]1CCCN1C(=O)C1=CC1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RHOC P08134 1/20 0.48
RHOA P61586 1/20 0.48
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
HTT P42858 2/20 0.46
MAPT P10636 1/20 0.46
NPC1 O15118 1/20 0.46
PABPC1 P11940 1/20 0.45
ALDH1A1 P00352 3/20 0.45
MAPK1 P28482 1/20 0.45
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
GAA P10253 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845300 0.84 CYP2C9 (0.54) RHOCRHOACYP2C9CYP2C19HTT
SCHEMBL844884 0.82 HTT (0.48) RHOCRHOACYP2C9CYP2C19HTT
SCHEMBL844934 0.82 RHOC (0.51) RHOCRHOACYP2C9CYP2C19HTT
SCHEMBL845181 0.81 MAPT (0.69) HTTMAPTPABPC1ALDH1A1
SCHEMBL845008 0.81 ALDH1A1 (0.54) CYP2C9CYP2C19HTTMAPTALDH1A1
SCHEMBL845255 0.81 CYP2C9 (0.47) RHOCRHOACYP2C9CYP2C19HTT
SCHEMBL845258 0.81 MAPK1 (0.60) CYP2C9CYP2C19HTTNPC1PABPC1
SCHEMBL845170 0.81 CYP2C9 (0.47) RHOCRHOACYP2C9CYP2C19HTT
SCHEMBL845541 0.80 RHOC (0.49) RHOCRHOACYP2C9CYP2C19HTT
SCHEMBL845443 0.80 CYP2C9 (0.47) RHOCRHOACYP2C9CYP2C19HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed