SCHEMBL8732014

SCHEMBL8732014

O=C(NCc1ccccc1)NC(Cc1ccccc1)C(O)CNCCc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 5/20 0.55
SLC6A11 P48066 1/20 0.55
EPHX1 P07099 1/20 0.54
ANPEP P15144 1/20 0.49
BCHE P06276 5/20 0.48
ATM Q13315 1/20 0.48
EPHX2 P34913 1/20 0.48
KMT2A Q03164 1/20 0.46
ALDH1A1 P00352 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8729415 0.90 BACE1 (0.67) BACE1SLC6A11ANPEPBCHEATM
SCHEMBL8955274 0.87 BACE1 (0.57) BACE1SLC6A11ANPEPBCHEATM
SCHEMBL7647681 0.87 L3MBTL1 (0.52) BACE1SLC6A11ANPEPBCHEATM
SCHEMBL8734455 0.87 L3MBTL1 (0.52) BACE1SLC6A11ANPEPBCHEATM
SCHEMBL3348148 0.85 BACE1 (0.54) BACE1SLC6A11ANPEPBCHE
SCHEMBL3348155 0.85 BACE1 (0.54) BACE1SLC6A11ANPEPBCHE
SCHEMBL8731471 0.85 BACE1 (0.55) BACE1SLC6A11ANPEPBCHEATM
SCHEMBL8734450 0.83 BCHE (0.68) BACE1SLC6A11ANPEPBCHEATM
SCHEMBL8731402 0.80 BACE1 (0.56) BACE1SLC6A11BCHE
SCHEMBL8734184 0.80 BCHE (0.58) BACE1SLC6A11BCHEATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5708004-A ENZYME INHIBITORS FOR TREATMENT OF AIDS MONSANTO COMPANY (US) 1998-01-13 US disclosed
US-5703076-A TREATING HIV, AIDS G. D. SEARLE & CO. (US) 1997-12-30 US disclosed
US-5698569-A Retroviral protease inhibitors G. D. SEARLE & CO. (US) 1997-12-16 US disclosed
US-5510349-A HUMAN IMMUNODEFICIENCY VIRUS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5510487-A TREATING HUMAN IMMUNODEFICIENCY VIRUS INFECTIONS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5510378-A Retroviral protease inhibitors G.D. SEARLE & CO. (US) 1996-04-23 US disclosed