SCHEMBL8423819

SCHEMBL8423819

NS(=O)(=O)c1ccccc1-n1nc(-c2ccc(Br)cc2)cc1-c1ccc(Cl)cc1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.51
PTGS1 P23219 3/20 0.48
MMP2 P08253 1/20 0.48
CYP2C9 P11712 1/20 0.44
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
USP8 P40818 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
SMPD1 P17405 1/20 0.41
MAPT P10636 1/20 0.40
MAPK9 P45984 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8424010 1.00 PTGS2 (0.51) PTGS2PTGS1MMP2CYP2C9CA1
SCHEMBL8421778 0.94 PTGS2 (0.56) PTGS2PTGS1CYP2C9MEN1KMT2A
SCHEMBL8422138 0.94 PTGS2 (0.56) PTGS2PTGS1MMP2CYP2C9CA1
SCHEMBL8733829 0.92 PTGS2 (0.54) PTGS2PTGS1MMP2CYP2C9MEN1
SCHEMBL8421736 0.90 PTGS2 (0.46) PTGS2PTGS1MMP2CYP2C9CA1
SCHEMBL8421816 0.90 PTGS2 (0.46) PTGS2PTGS1MMP2CYP2C9CA1
SCHEMBL8423767 0.90 PTGS2 (0.52) PTGS2PTGS1CYP2C9MEN1KMT2A
SCHEMBL8422286 0.90 PTGS2 (0.52) PTGS2PTGS1CYP2C9MEN1KMT2A
SCHEMBL8424076 0.89 CYP2C9 (0.57) PTGS2PTGS1CYP2C9CA1CA2
SCHEMBL8423901 0.89 PTGS2 (0.51) PTGS2PTGS1MMP2CYP2C9MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5908852-A 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation G. D. SEARLE & CO. (US) 1999-06-01 US disclosed