SCHEMBL8733910

SCHEMBL8733910

NCCCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCN(c4ncccn4)CC3)c(C(F)(F)F)c21

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.55
ALDH1A1 P00352 7/20 0.43
HPGD P15428 6/20 0.43
HSD17B10 Q99714 5/20 0.43
ADRA2B P18089 1/20 0.42
MAPK1 P28482 1/20 0.42
DRD3 P35462 1/20 0.42
PMP22 Q01453 1/20 0.42
PIK3CG P48736 1/20 0.41
ALB P02768 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
AADAT Q8N5Z0 2/20 0.40
TUBB4A P04350 1/20 0.40
POLB P06746 1/20 0.40
TUBB P07437 1/20 0.40
TUBA3C P0DPH7 1/20 0.40
TUBA1B P68363 1/20 0.40
TUBA4A P68366 1/20 0.40
TUBB4B P68371 1/20 0.40
TUBB3 Q13509 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8059291 0.95 KDM4E (0.62) KDM4EALDH1A1HPGDHSD17B10ADRA2B
SCHEMBL8057366 0.90 KDM4E (0.53) KDM4EALDH1A1HPGDHSD17B10ADRA2B
SCHEMBL8057434 0.86 KDM4E (0.50) KDM4EALDH1A1HPGDHSD17B10ADRA2B
SCHEMBL8730261 0.86 KDM4E (0.47) KDM4EALDH1A1HPGDHSD17B10ADRA2B
SCHEMBL8736312 0.86 KDM4E (0.55) KDM4EALDH1A1HPGDHSD17B10ADRA2B
SCHEMBL8064088 0.85 KDM4E (0.58) KDM4EALDH1A1HPGDHSD17B10ADRA2B
SCHEMBL8058583 0.84 KDM4E (0.48) KDM4EALDH1A1HPGDHSD17B10ADRA2B
SCHEMBL8064229 0.82 KDM4E (0.48) KDM4EALDH1A1HPGDHSD17B10ADRA2B
SCHEMBL8058512 0.82 ALDH1A1 (0.52) KDM4EALDH1A1HPGDHSD17B10PIK3CG
SCHEMBL8059277 0.81 KDM4E (0.49) KDM4EALDH1A1HPGDHSD17B10DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0878194-A1 REMEDIES OR PREVENTIVES FOR AIDS SANKYO COMPANY LIMITED (JP) 1998-11-18 EP disclosed