Cambendazole

Cambendazole

SCHEMBL8734398

CC(C)OC(=O)Nc1ccc2[nH]c(-c3cscn3)nc2c1.c1ccc2[nH]c(-c3cscn3)nc2c1

nearest known ligand 0.80

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
METAP1 P53582 6/20 0.57
METAP2 P50579 5/20 0.57
SMN1; SMN2 Q16637 5/20 0.57
KDM4E B2RXH2 5/20 0.57
TP53 P04637 4/20 0.57
NPC1 O15118 3/20 0.57
RAB9A P51151 3/20 0.57
CYP1A2 P05177 1/20 0.57
CYP3A4 P08684 1/20 0.57
ADORA3 P0DMS8 1/20 0.57
CYP2D6 P10635 1/20 0.57
TSHR P16473 1/20 0.57
CYP2C19 P33261 1/20 0.57
FKBP1A P62942 1/20 0.57
HIF1A Q16665 1/20 0.57
TDP1 Q9NUW8 1/20 0.57
HDAC6 Q9UBN7 1/20 0.57
MAPT P10636 3/20 0.43
RXFP1 Q9HBX9 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cambendazole SCHEMBL44000 0.95 METAP1 (0.48) METAP1METAP2SMN1; SMN2KDM4ETP53
Cambendazole SCHEMBL29409263 0.95 METAP1 (0.48) METAP1METAP2SMN1; SMN2KDM4ETP53
Cambendazole SCHEMBL2895694 0.89 METAP1 (0.55) METAP1METAP2SMN1; SMN2KDM4ETP53
Diethenofencarb SCHEMBL9055860 0.89 HPSE (0.51) METAP1METAP2SMN1; SMN2KDM4ETP53
SCHEMBL3500748 0.85 METAP1 (0.52) METAP1METAP2SMN1; SMN2KDM4ETP53
Mebendazole SCHEMBL2406875 0.84 METAP1 (0.54) METAP1METAP2SMN1; SMN2KDM4ETP53
SCHEMBL4366074 0.81 METAP1 (0.50) METAP1METAP2SMN1; SMN2KDM4ETP53
SCHEMBL4367982 0.81 METAP1 (0.50) METAP1METAP2SMN1; SMN2KDM4ETP53
SCHEMBL11208569 0.79 METAP1 (0.55) METAP1METAP2SMN1; SMN2KDM4ETP53
SCHEMBL4367695 0.79 METAP1 (0.48) METAP1METAP2SMN1; SMN2KDM4ETP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3247701-B1 ANTHELMINTIC COMPOUNDS, COMPOSITIONS AND METHOD OF USING THEREOF BOEHRINGER INGELHEIM ANIMAL HEALTH USA INC (US) 2021-09-22 EP disclosed
US-10597364-B2 Anthelmintic compounds, compositions and method of using thereof Boehringer Ingelheim Animal Health USA Inc. (US) 2020-03-24 US disclosed
US-20180009754-A1 ANTHELMINTIC COMPOUNDS, COMPOSITIONS AND METHOD OF USING THEREOF MERIAL, INC. (US) 2018-01-11 US disclosed
EP-3247701-A1 ANTHELMINTIC COMPOUNDS, COMPOSITIONS AND METHOD OF USING THEREOF Merial, Inc. (US) 2017-11-29 EP disclosed
WO-2016118638-A1 ANTHELMINTIC COMPOUNDS, COMPOSITIONS AND METHOD OF USING THEREOF MERIAL INC. (US) 2016-07-28 WO disclosed
EP-0710105-A4 SYNERGISTIC ANTHELMINTIC COMPOSITIONS UNIV AUSTRALIAN (AU) 1998-06-10 EP disclosed
EP-0710105-A1 SYNERGISTIC ANTHELMINTIC COMPOSITIONS THE AUSTRALIAN NATIONAL UNIVERSITY (AU) 1996-05-08 EP disclosed
WO-1994028887-A1 SYNERGISTIC ANTHELMINTIC COMPOSITIONS THE AUSTRALIAN NATIONAL UNIVERSITY (AU) 1994-12-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10597364-B2 Anthelmintic compounds, compositions and method of using thereof CYP8B1, CYP2C8, CYP2B6 METAP1 1022/4885METAP2 795/4885SMN1; SMN2 4838/4885
US-20180009754-A1 ANTHELMINTIC COMPOUNDS, COMPOSITIONS AND METHOD OF USING THEREOF CYP8B1, CYP2C8, CYP2B6 METAP1 1022/4885METAP2 795/4885SMN1; SMN2 4838/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.