SCHEMBL8735880

SCHEMBL8735880

O=C(O)c1cn(Cc2ccccn2)c2c(OC(F)F)c(F)c(F)cc2c1=O

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.49
CHRM1 P11229 2/20 0.41
SLC22A12 Q96S37 1/20 0.41
TOP1 P11387 6/20 0.41
TOP2A P11388 2/20 0.37
TOP2B Q02880 2/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.36
GSK3B P49841 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8736423 0.89 STAT3 (0.43) KDM4EALDH1A1
SCHEMBL8736415 0.86 CHRM1 (0.53) CHRM1TOP1MAPT
SCHEMBL8735563 0.80 KDM4E (0.51) KDM4EALDH1A1
SCHEMBL8733989 0.79 KDM4E (0.47) KDM4ECHRM1TOP1TOP2ATOP2B
SCHEMBL8733567 0.77 KDM4E (0.48) KDM4ECHRM1TOP1ALDH1A1
SCHEMBL8731834 0.74 KDM4E (0.43) KDM4ETOP1TOP2ATOP2BALDH1A1
SCHEMBL8735858 0.73 KDM4E (0.40) KDM4ETOP1TOP2ATOP2BALDH1A1
SCHEMBL8736445 0.72 KDM4E (0.50) KDM4ETOP1ALDH1A1
SCHEMBL21787284 0.71 TOP1 (0.68) CHRM1TOP1
SCHEMBL7009985 0.71 CHRM1 (0.61) KDM4ECHRM1TOP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0878194-A1 REMEDIES OR PREVENTIVES FOR AIDS SANKYO COMPANY LIMITED (JP) 1998-11-18 EP disclosed
US-5688791-A COMPOUNDS FOR TREATMENNT OF VIRAL DISEASES SUCH AS AIDS UBE INDUSTRIES, LTD. (JP) 1997-11-18 US disclosed
US-5519016-A Aryl group- or aromatic heterocyclic group-substituted aminoquinolone derivatives and anti-HIV agent UBE INDUSTRIES, LTD. (JP) 1996-05-21 US disclosed
EP-0572259-A1 Aminoquinolone derivatives as anti-HIV agents UBE INDUSTRIES, LTD. (JP) 1993-12-01 EP disclosed