SCHEMBL8736649

SCHEMBL8736649

CC1CC(C)C(C)(C)c2ccc(CC#Cc3ccc(C(=O)Nc4ccc(O)cc4)cc3)cc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP26A1 O43174 4/20 0.38
CYP26B1 Q9NR63 2/20 0.38
NQO2 P16083 2/20 0.36
SNCA P37840 1/20 0.36
DEGS1 O15121 2/20 0.35
KMT2A Q03164 7/20 0.35
MEN1 O00255 6/20 0.35
POLB P06746 2/20 0.35
USP2 O75604 1/20 0.35
HIF1A Q16665 3/20 0.34
EPAS1 Q99814 3/20 0.34
CYP3A4 P08684 2/20 0.34
RARA P10276 2/20 0.34
RARB P10826 2/20 0.34
RARG P13631 2/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7746394 0.80 CYP26A1 (0.57) CYP26A1CYP26B1NQO2SNCAKMT2A
SCHEMBL10439232 0.66 MMP2 (0.48) NQO2SNCADEGS1KMT2AMEN1
SCHEMBL6340122 0.66 BACE1 (0.37) CYP26A1CYP26B1SNCADEGS1KMT2A
SCHEMBL7746406 0.65 CYP26A1 (0.53) CYP26A1CYP26B1KMT2AMEN1CYP3A4
SCHEMBL6873454 0.64 CYP26A1 (0.54) CYP26A1CYP26B1NQO2SNCADEGS1
SCHEMBL7928437 0.64 RARB (0.55) CYP26A1CYP26B1CYP3A4RARARARB
SCHEMBL7746076 0.64 CYP26A1 (0.48) CYP26A1CYP26B1CYP3A4RARARARB
SCHEMBL7752015 0.63 CYP26A1 (0.51) CYP26A1CYP26B1KMT2AMEN1CYP3A4
SCHEMBL10439244 0.63 DEGS1 (0.69) NQO2SNCADEGS1KMT2AMEN1
SCHEMBL10439472 0.63 DEGS1 (0.46) NQO2SNCADEGS1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832057-A1 DIAROMATIC PROPYNYL OR DIENYL COMPOUNDS CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (C.I.R.D. GALDERMA) (FR) 1998-04-01 EP claimed
WO-1997033856-A1 DIAROMATIC PROPYNYL OR DIENYL COMPOUNDS CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (C.I.R.D. GALDERMA) (FR) 1997-09-18 WO claimed