SCHEMBL8743221

SCHEMBL8743221

[CH2]COC(=O)c1ccc(Br)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.56
NPC1 O15118 1/20 0.56
RAB9A P51151 1/20 0.56
KDM4E B2RXH2 4/20 0.53
LMNA P02545 2/20 0.53
MAPT P10636 4/20 0.50
KMT2A Q03164 2/20 0.50
ALDH1A1 P00352 2/20 0.50
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
POLB P06746 1/20 0.47
MEN1 O00255 1/20 0.47
GSK3B P49841 2/20 0.47
CHRNB2 P17787 1/20 0.45
CHRNA7 P36544 1/20 0.45
CHRNA4 P43681 1/20 0.45
NHERF1 O14745 1/20 0.45
OGG1 O15527 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6964934 0.79 GAA (0.53) NPC1RAB9AKDM4ELMNAMAPT
SCHEMBL11320755 0.79 CA1 (0.57) HPGDNPC1RAB9AKDM4EMAPT
SCHEMBL3022388 0.79 MAPT (0.51) HPGDNPC1RAB9AKDM4ELMNA
SCHEMBL274513 0.79 CA1 (0.68) HPGDNPC1RAB9AKDM4ELMNA
SCHEMBL8742866 0.79 TDP1 (0.57) HPGDNPC1RAB9ALMNAMAPT
SCHEMBL22995612 0.79 HPGD (0.56) HPGDNPC1RAB9AKDM4ELMNA
SCHEMBL4433115 0.79 SNCA (0.58) HPGDNPC1RAB9AKDM4ELMNA
SCHEMBL112532 0.78 TDP1 (0.63) HPGDNPC1RAB9AKDM4ELMNA
SCHEMBL20607027 0.78 HPGD (0.54) HPGDNPC1RAB9AKDM4ELMNA
SCHEMBL2989285 0.78 CA12 (0.66) HPGDNPC1RAB9AKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0751113-A1 Optically active phenol derivatives and preparation thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-01-02 EP disclosed
US-5420363-A Catalytic reaction of phenol with secondary carbinol for enantiomorphs TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-05-30 US disclosed
US-5354913-A Chemical intermediates for drugs or drugs as thromboxane, prostaglandin antagonist, lipoxygenase enzyme inhibitor, antioxidants TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-10-11 US disclosed
EP-0582382-A2 Optically active phenol derivatives and preparation thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-02-09 EP disclosed