SCHEMBL8743644

SCHEMBL8743644

[CH2]COP(Oc1ccccc1)Oc1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 3/20 0.36
TSHR P16473 1/20 0.36
KCNA3 P22001 1/20 0.36
CA4 P22748 1/20 0.33
KMT2A Q03164 1/20 0.32
APP P05067 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32
ALDH1A1 P00352 1/20 0.32
RECQL P46063 1/20 0.32
ALOX15 P16050 1/20 0.31
CA5A P35218 1/20 0.30
CA5B Q9Y2D0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14354354 0.81 KCNA3 (0.44) LTA4HTSHRKCNA3CA4KMT2A
SCHEMBL25813074 0.77 KCNA3 (0.46) LTA4HTSHRKCNA3TAAR1ALDH1A1
SCHEMBL28530483 0.77 ALDH1A1 (0.41) LTA4HTSHRKCNA3CA4KMT2A
SCHEMBL443626 0.77 LTA4H (0.43) LTA4HTSHRKCNA3CA4
SCHEMBL28017927 0.77 LTA4H (0.50) LTA4HTSHRKCNA3CA4KMT2A
SCHEMBL13289 0.77 LTA4H (0.50) LTA4HTSHRKCNA3CA4KMT2A
SCHEMBL250539 0.77 CYP3A4 (0.36) LTA4HTSHRKCNA3KMT2AALDH1A1
SCHEMBL5929542 0.76 TSHR (0.46) TSHRKMT2AAPPALDH1A1
SCHEMBL11871889 0.75 LTA4H (0.47) LTA4HTSHRKCNA3CA4KMT2A
SCHEMBL3009883 0.75 LTA4H (0.47) LTA4HTSHRKCNA3CA4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0646146-B1 IMPROVED PROCESS FOR PREPARING EXTENDED CHAIN POLYESTERS AND BLOCK OR GRAFT COPOLYESTERS ALLIED SIGNAL INC (US) 1997-11-12 EP disclosed
EP-0651774-B1 PROCESS FOR PREPARING CHAIN EXTENDED POLYMERS AND GRAFT AND BLOCK COPOLYMERS ALLIED SIGNAL INC (US) 1997-01-08 EP disclosed
EP-0651774-A1 PROCESS FOR PREPARING CHAIN EXTENDED POLYMERS AND GRAFT AND BLOCK COPOLYMERS. ALLIED SIGNAL INC (US) 1995-05-10 EP disclosed
EP-0646146-A1 IMPROVED PROCESS FOR PREPARING EXTENDED CHAIN POLYESTERS AND BLOCK OR GRAFT COPOLYESTERS AlliedSignal Inc. (US) 1995-04-05 EP disclosed
US-5389721-A Using phosphorous(III)-containing chain extension reagents; heating; using no catalytic substances which contain elements from groups VA and VIA of the periodic table ALLIEDSIGNAL INC. (US) 1995-02-14 US disclosed
US-5326830-A Heterocyclic nitrogen-trivalent phosphorous compounds ALLIEDSIGNAL INC. (US) 1994-07-05 US disclosed
WO-1994010242-A1 NUCLEATING SYSTEM FOR POLYESTERS AND ARTICLES FORMED THEREFROM ALLIED-SIGNAL INC. (US) 1994-05-11 WO disclosed
WO-1994002537-A1 PROCESS FOR PREPARING CHAIN EXTENDED POLYMERS AND GRAFT AND BLOCK COPOLYMERS ALLIED-SIGNAL INC. (US) 1994-02-03 WO disclosed
WO-1993025601-A1 IMPROVED PROCESS FOR PREPARING EXTENDED CHAIN POLYESTERS AND BLOCK OR GRAFT COPOLYESTERS ALLIED-SIGNAL INC. (US) 1993-12-23 WO disclosed
US-4963311-A GRAFTING A PHOSPHITE-MODIFIED POLYESTER BASED ON A CARBO DIACID AND A CARBO OR ACYCLIC GLYCOL TO A NYLON; SPINNING AND DRAWING ALLIED-SIGNAL (US) 1990-10-16 US disclosed
US-4568720-A WITH PHOSPHITE COMPOUND ALLIED CHEMICAL CORPORATION (US) 1986-02-04 US disclosed