SCHEMBL874382

SCHEMBL874382

O=c1nn[nH]c2cc(OC(F)(F)F)ccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.48
TRPA1 O75762 5/20 0.47
SCN5A Q14524 1/20 0.47
SCN9A Q15858 1/20 0.47
KDM4E B2RXH2 2/20 0.43
CRHBP P24387 1/20 0.43
CRHR2 Q13324 1/20 0.43
CES1 P23141 1/20 0.43
METAP2 P50579 1/20 0.41
NOTUM Q6P988 1/20 0.38
GSK3B P49841 2/20 0.38
ABL1 P00519 1/20 0.38
POLB P06746 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
GAA P10253 1/20 0.37
KMT2A Q03164 1/20 0.37
RUNX1 Q01196 1/20 0.36
CBFB Q13951 1/20 0.36
TRPV1 Q8NER1 1/20 0.36
GPR3 P46089 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16178955 0.78 KIF11 (0.45) KIF11TRPA1SCN5ASCN9ACES1
SCHEMBL874384 0.76 CES1 (0.43) KIF11TRPA1SCN5ASCN9AKDM4E
SCHEMBL203008 0.74 KIF11 (0.41) KIF11TRPA1SCN5ASCN9AKDM4E
SCHEMBL12515210 0.72 TRPA1 (0.52) KIF11TRPA1SCN5ASCN9AKDM4E
SCHEMBL2856373 0.71 TRPA1 (0.51) KIF11TRPA1SCN5ASCN9AGSK3B
SCHEMBL10883616 0.70 DAO (0.47) KDM4EGSK3BKMT2A
SCHEMBL10987571 0.70 JAK2 (0.50) METAP2GSK3BABL1
SCHEMBL3119854 0.70 KIF11 (0.64) KIF11TRPA1SCN5ASCN9AKDM4E
SCHEMBL21145515 0.69 HSD17B10 (0.59) KIF11TRPA1SCN5ASCN9AKDM4E
SCHEMBL7033184 0.69 KIF11 (0.58) KIF11TRPA1SCN5ASCN9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2619179-A1 MATRIX METALLOPROTEINASE INHIBITORS Ranbaxy Laboratories Limited (IN) 2013-07-31 EP disclosed
WO-2012038944-A1 MATRIX METALLOPROTEINASE INHIBITORS RANBAXY LABORATORIES LIMITED (IN) 2012-03-29 WO disclosed