SCHEMBL8744009

SCHEMBL8744009

CCC1CCC(=Nc2cccc(C)c2)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.38
KMT2A Q03164 4/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CRHBP P24387 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTT P42858 1/20 0.38
CRHR2 Q13324 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HTR3E A5X5Y0 2/20 0.38
HTR3B O95264 2/20 0.38
HTR3A P46098 2/20 0.38
HTR3D Q70Z44 2/20 0.38
HTR3C Q8WXA8 2/20 0.38
MAPT P10636 2/20 0.36
NPC1 O15118 1/20 0.34
NSD2 O96028 1/20 0.34
CASP3 P42574 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8743971 0.82 HTR3E (0.41) MEN1KMT2ASMN1; SMN2CYP3A4CYP2D6
SCHEMBL8744092 0.82 MAPT (0.35) SMN1; SMN2CYP2C19HTTMAPTTDP1
SCHEMBL8743991 0.81 HTR3E (0.40) MEN1KMT2ASMN1; SMN2CYP3A4CYP2D6
SCHEMBL8743959 0.81 HTR3E (0.43) MEN1KMT2ASMN1; SMN2CYP3A4CYP2D6
SCHEMBL8743966 0.80 ALDH1A1 (0.33) SMN1; SMN2HTR3EHTR3BHTR3AHTR3D
SCHEMBL8744074 0.78 HTR3E (0.38) MEN1KMT2ASMN1; SMN2CYP3A4CYP2D6
SCHEMBL16620267 0.77 SMN1; SMN2 (0.38) MEN1KMT2ASMN1; SMN2CYP3A4CYP2D6
SCHEMBL8743975 0.76 HTR3E (0.44) MEN1KMT2ASMN1; SMN2CYP3A4CYP2D6
SCHEMBL8743916 0.75 ALDH1A1 (0.38) MEN1KMT2ACYP3A4HTTNPSR1
SCHEMBL18395323 0.75 MAPT (0.37) MEN1KMT2ASMN1; SMN2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5618980-A DEHYDROGENATING N-CYCLOHEXYLIDENEAMINO COMPOUND IN PRESENCE OF HYDROGEN TRANSFER CATALYST AND HYDROGEN ACCEPTOR AND ALKALI OR ALKALINE EARTH METAL COMPOUND COCATALYST MITSUI TOATSU CHEMICALS, INC. (JP) 1997-04-08 US disclosed
EP-0588060-B1 Method for preparing aromatic secondary amino compound MITSUI TOATSU CHEMICALS (JP) 1997-04-02 EP disclosed
EP-0753505-A2 Method for preparing aromatic secondary amino compound MITSUI TOATSU CHEMICALS, Inc. (JP) 1997-01-15 EP disclosed
US-5536878-A HYDROGEN ACCEPTOR MITSUI TOATSU CHEMICALS, INC. (JP) 1996-07-16 US disclosed
US-5382690-A Method for preparing aromatic secondary amino compound MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1995-01-17 US disclosed
EP-0588060-A2 Method for preparing aromatic secondary amino compound MITSUI TOATSU CHEMICALS, Inc. (JP) 1994-03-23 EP disclosed