SCHEMBL874458

SCHEMBL874458

O=C1NC(=O)C2(N1)C1=C(C=CCO1)Oc1ccccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 1/20 0.42
CYP2C9 P11712 2/20 0.38
CACNA1F O60840 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
HTR2A P28223 1/20 0.38
HRH1 P35367 1/20 0.38
SCN1A P35498 1/20 0.38
SCN4A P35499 1/20 0.38
BLM P54132 1/20 0.38
PMP22 Q01453 1/20 0.38
CACNA1D Q01668 1/20 0.38
KCNH2 Q12809 1/20 0.38
CACNA1S Q13698 1/20 0.38
CACNA1C Q13936 1/20 0.38
SCN5A Q14524 1/20 0.38
SCN2A Q99250 1/20 0.38
SCN3A Q9NY46 1/20 0.38
TSHR P16473 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL877138 0.76 ITGA4 (0.65) ITGA4CYP2C9CACNA1FALDH1A1MAPT
SCHEMBL23998300 0.65 AKR1B1 (0.67) ITGA4CYP2C9CACNA1FALDH1A1MAPT
SCHEMBL23178755 0.65 ITGA4 (0.45) ITGA4CYP2C9CACNA1FALDH1A1MAPT
SCHEMBL10606071 0.61 TSHR (0.49) ITGA4TSHRTDP1AKR1B1
SCHEMBL31195728 0.61 ITGA4 (1.00) ITGA4CYP2C9CACNA1FALDH1A1MAPT
SCHEMBL9810959 0.61 ITGA4 (1.00) ITGA4CYP2C9CACNA1FALDH1A1MAPT
SCHEMBL23178807 0.61 ITGA4 (0.40) ITGA4CYP2C9CACNA1FALDH1A1MAPT
SCHEMBL30297506 0.61 TSHR (0.55) MAPTTSHRTDP1AKR1B1AKR1A1
SCHEMBL3035791 0.60 ITGA4 (0.63) ITGA4CYP2C9CACNA1FALDH1A1MAPT
SCHEMBL7876513 0.60 AKR1B1 (0.65) MAPTTSHRTDP1AKR1B1AKR1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012040641-A2 COMPOUNDS FOR TREATING NEURODEGENERATIVE DISEASES ARRAY BIOPHARMA INC. (US) 2012-03-29 WO disclosed