SCHEMBL23178807

SCHEMBL23178807

C=CC1=C(/C=C\C)Oc2ccccc2[C@]12NC(=O)NC2=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 1/20 0.40
CYP2C9 P11712 2/20 0.36
CACNA1F O60840 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
HTR2A P28223 1/20 0.36
HRH1 P35367 1/20 0.36
SCN1A P35498 1/20 0.36
SCN4A P35499 1/20 0.36
BLM P54132 1/20 0.36
PMP22 Q01453 1/20 0.36
CACNA1D Q01668 1/20 0.36
KCNH2 Q12809 1/20 0.36
CACNA1S Q13698 1/20 0.36
CACNA1C Q13936 1/20 0.36
SCN5A Q14524 1/20 0.36
SCN2A Q99250 1/20 0.36
SCN3A Q9NY46 1/20 0.36
CRHBP P24387 1/20 0.35
CRHR2 Q13324 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23178755 0.89 ITGA4 (0.45) ITGA4CYP2C9CACNA1FALDH1A1MAPT
SCHEMBL877138 0.74 ITGA4 (0.65) ITGA4CYP2C9CACNA1FALDH1A1MAPT
SCHEMBL24877020 0.72 PDK2 (0.32)
SCHEMBL23697575 0.67 FTO (0.35) ALDH1A1MAPTBLM
SCHEMBL23874319 0.65 NTSR1 (0.35) ALDH1A1
SCHEMBL24487581 0.64 PDK2 (0.34)
SCHEMBL23008568 0.64 PDK2 (0.32)
SCHEMBL19886292 0.64 KDM4E (0.39) ALDH1A1MAPT
SCHEMBL24979979 0.63 CHRM3 (0.35)
SCHEMBL22110666 0.62 FTO (0.62) CYP2C9ALDH1A1MAPTBLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021061763-A1 ALDOKETO REDUCTASE INHIBITORS AND USES THEREOF CASE WESTERN RESERVE UNIVERSITY (US) 2021-04-01 WO disclosed