SCHEMBL8744815

SCHEMBL8744815

CCOC(=O)CNC(=O)Cc1ccc(Cl)cc1Cl

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.56
ERCC1 P07992 5/20 0.52
ERCC4 Q92889 5/20 0.52
KMT2A Q03164 2/20 0.52
ALDH1A1 P00352 2/20 0.52
HTT P42858 2/20 0.52
KDM4E B2RXH2 1/20 0.52
MEN1 O00255 1/20 0.52
THRB P10828 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
TDP1 Q9NUW8 1/20 0.50
P2RX7 Q99572 5/20 0.49
NPC1 O15118 2/20 0.48
RAB9A P51151 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13310056 0.87 GAA (0.54) GAAKMT2AALDH1A1HTTMEN1
SCHEMBL13190848 0.85 PPID (0.56) GAAALDH1A1HTTTDP1P2RX7
SCHEMBL31441299 0.84 KMT2A (0.57) GAAERCC1ERCC4KMT2AALDH1A1
SCHEMBL707398 0.84 KMT2A (0.57) GAAERCC1ERCC4KMT2AALDH1A1
SCHEMBL3448919 0.83 NPC1 (0.54) GAAKMT2AALDH1A1HTTMEN1
SCHEMBL8424664 0.81 ERCC1 (0.61) ERCC1ERCC4KMT2AP2RX7NPC1
SCHEMBL15211291 0.80 PPARD (0.45) GAAKMT2AALDH1A1HTTKDM4E
SCHEMBL8744740 0.80 ERCC1 (0.59) ERCC1ERCC4KMT2AALDH1A1P2RX7
SCHEMBL10900050 0.78 ALDH1A1 (0.45) GAAERCC1ERCC4KMT2AALDH1A1
SCHEMBL28224249 0.77 SMN1; SMN2 (0.58) ERCC1ERCC4KMT2AALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0456063-B1 1-H-3-aryl-pyrrolidin-2,4-dion-derivatives BAYER AG (DE) 1997-01-22 EP disclosed
US-5258527-A Insecticidal, acaricidal and herbicidal 1-H-3-aryl-pyrrolidine-2,4-dione derivatives BAYER AKTIENGESELLSCHAFT (DE) 1993-11-02 US disclosed
EP-0456063-A2 1-H-3-aryl-pyrrolidin-2,4-dion-derivatives BAYER AG (DE) 1991-11-13 EP disclosed