SCHEMBL8745753

SCHEMBL8745753

COc1ccc2c(C)c(CCO)c(=O)oc2c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 0.61
GAA P10253 2/20 0.61
TP53 P04637 1/20 0.61
KDM4E B2RXH2 10/20 0.60
ALDH1A1 P00352 9/20 0.60
HPGD P15428 6/20 0.60
HSD17B10 Q99714 5/20 0.60
MAPT P10636 5/20 0.60
THRB P10828 1/20 0.60
RAB9A P51151 5/20 0.58
NPC1 O15118 4/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
POLB P06746 1/20 0.55
STAT1 P42224 1/20 0.55
HSD17B3 P37058 1/20 0.54
STS P08842 1/20 0.54
ACHE P22303 1/20 0.53
MAOB P27338 1/20 0.53
TSHR P16473 1/20 0.53
LMNA P02545 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29699265 0.86 KDM4E (0.60) NQO1GAATP53KDM4EALDH1A1
SCHEMBL18766190 0.86 KDM4E (0.60) NQO1GAATP53KDM4EALDH1A1
SCHEMBL24627780 0.83 MAPT (0.72) GAATP53KDM4EALDH1A1HPGD
SCHEMBL7141692 0.82 KDM4E (0.55) NQO1GAATP53KDM4EALDH1A1
SCHEMBL29944843 0.82 KDM4E (0.55) NQO1GAATP53KDM4EALDH1A1
Ocimarin SCHEMBL23752453 0.82 HSD17B3 (0.79) NQO1GAATP53KDM4EALDH1A1
SCHEMBL237672 0.81 KDM4E (0.54) NQO1GAATP53KDM4EALDH1A1
SCHEMBL8745770 0.81 ALDH1A1 (0.57) NQO1GAATP53KDM4EALDH1A1
SCHEMBL22733326 0.81 KDM4E (0.77) GAAKDM4EALDH1A1HPGDHSD17B10
SCHEMBL8745776 0.81 NQO1 (0.59) NQO1TP53KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0663911-B1 BENZOPYRANONES, METHOD OF PREPARING THEM AND THEIR USE SCHWABE WILLMAR GMBH & CO (DE) 1997-02-05 EP disclosed
US-5550129-A THERAPY FOR NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS WILLMAR SCHWABE GMBH & CO. (DE) 1996-08-27 US disclosed
EP-0663911-A1 BENZOPYRANONES, METHOD OF PREPARING THEM AND THEIR USE. SCHWABE WILLMAR GMBH & CO (DE) 1995-07-26 EP disclosed
WO-1994008985-A1 BENZOPYRANONES, METHOD OF PREPARING THEM AND THEIR USE DR. WILLMAR SCHWABE GMBH & CO. (DE) 1994-04-28 WO disclosed