SCHEMBL8747014

SCHEMBL8747014

COc1cc2c(cc1O)C(C1(c3ccc(OC(F)(F)F)cc3)CCC1)N(C)CC2

nearest known ligand 0.60

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.60
DRD1 P21728 4/20 0.60
CYP2D6 P10635 1/20 0.60
KCNH2 Q12809 1/20 0.43
MAOA P21397 1/20 0.43
PDE4B Q07343 1/20 0.41
PDE4D Q08499 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL8747231 0.96 DRD2 (0.56) DRD2DRD1CYP2D6KCNH2MAOA
SCHEMBL8747234 0.87 CYP2D6 (0.46) DRD2DRD1CYP2D6KCNH2PDE4B
SCHEMBL8747012 0.86 DRD1 (0.50) DRD2DRD1MAOA
SCHEMBL8747191 0.85 DRD1 (0.56) DRD2DRD1KCNH2MAOA
SCHEMBL8747029 0.84 DRD1 (0.50) DRD2DRD1MAOA
SCHEMBL8747267 0.83 CHRNA7 (0.46) DRD2DRD1CYP2D6
SCHEMBL8747299 0.83 DRD1 (0.47) DRD2DRD1KCNH2MAOA
SCHEMBL8747074 0.83 DRD1 (0.49) DRD2DRD1MAOA
SCHEMBL8747084 0.83 MAOA (0.45) DRD2DRD1KCNH2MAOA
Hydrochloric Acid SCHEMBL8747265 0.83 CHRNA7 (0.46) DRD2DRD1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618900-B1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS KNOLL AG (DE) 1997-03-12 EP disclosed
US-5519034-A ANALGESICS THE BOOTS COMPANY PLC (GB) 1996-05-21 US disclosed