Iodide

Iodide

SCHEMBL8747174

COc1cc2c(cc1OC)C(C1(c3ccccc3C#N)CCC1)=[N+](C)CC2.[I-]

nearest known ligand 0.39

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHRM1CHRM3CHRNA1CHRNB1CHRNDCHRNECHRNG

The experimentally established mechanism targets of Iodide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE known ✓ P22303 4/20 0.39
GAA P10253 1/20 0.38
ALOX12 P18054 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HIF1A Q16665 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
MAOA P21397 2/20 0.33
GLA P06280 1/20 0.33
PDGFRB P09619 1/20 0.32
PGR P06401 1/20 0.32
AR P10275 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA4 P22748 1/20 0.32
CA6 P23280 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8747302 0.77 RAD52 (0.43) GAAALOX12HTTSMN1; SMN2HIF1A
Iodide SCHEMBL8747182 0.74 CHRNA7 (0.40) ACHE
Iodide SCHEMBL7064042 0.65 ACHE (0.50) ACHEHIF1AMEN1KMT2AKDM4E
SCHEMBL8746994 0.64 MAOA (0.44) MEN1KMT2AKDM4EALDH1A1MAOA
Iodide SCHEMBL7060534 0.64 ACHE (0.54) ACHEGAAHIF1AMEN1KMT2A
Iodide SCHEMBL27348744 0.63 MAOA (0.44) MEN1KMT2AKDM4EALDH1A1MAOA
SCHEMBL27348743 0.63 MEN1 (0.41) MEN1KMT2AKDM4EALDH1A1MAOA
SCHEMBL19055622 0.62 ACHE (0.55) ACHEGAAHIF1AMEN1KMT2A
Iodide SCHEMBL10705028 0.58 ACHE (0.50) ACHEGAAHIF1AMEN1KMT2A
SCHEMBL14131507 0.57 ACHE (0.49) ACHEKDM4EGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618900-B1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS KNOLL AG (DE) 1997-03-12 EP disclosed
US-5519034-A ANALGESICS THE BOOTS COMPANY PLC (GB) 1996-05-21 US disclosed
EP-0618900-A1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS. BOOTS CO PLC (GB) 1994-10-12 EP disclosed
WO-1993013073-A1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS THE BOOTS COMPANY PLC (GB) 1993-07-08 WO disclosed