SCHEMBL8747190

SCHEMBL8747190

CN1CCc2ccc(O)cc2C1C1(c2ccc(Cl)cc2)CCC1

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 1/20 0.58
SLC6A2 P23975 2/20 0.42
SLC6A4 P31645 2/20 0.42
SLC6A3 Q01959 2/20 0.42
DRD1 P21728 11/20 0.41
HTR2A P28223 1/20 0.41
DRD2 P14416 8/20 0.41
DRD5 P21918 7/20 0.41
DRD3 P35462 7/20 0.41
DRD4 P21917 5/20 0.41
ESR1 P03372 2/20 0.41
ESR2 Q92731 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8747213 0.89 DRD1 (0.49) SLC6A9DRD1HTR2ADRD2DRD5
Hydrochloric Acid SCHEMBL8747194 0.88 DRD1 (0.50) SLC6A9DRD1HTR2ADRD2DRD5
SCHEMBL8747405 0.87 MAOA (0.47) SLC6A9DRD1DRD2DRD5DRD3
Bromide SCHEMBL8747099 0.86 MAOA (0.46) SLC6A9DRD1DRD2DRD3DRD4
SCHEMBL8747142 0.85 DRD1 (0.53) DRD1DRD2DRD5DRD4
SCHEMBL8747027 0.85 MAOA (0.47) SLC6A9DRD1DRD2DRD5DRD3
SCHEMBL8747031 0.84 MAOA (0.46) SLC6A9DRD1DRD2DRD5DRD3
SCHEMBL8747078 0.84 DRD1 (0.44) SLC6A9DRD1HTR2ADRD2DRD5
SCHEMBL8747307 0.83 DRD1 (0.41) SLC6A9DRD1DRD2DRD5DRD4
Bromide SCHEMBL8747367 0.83 DRD1 (0.43) SLC6A9DRD1HTR2ADRD2DRD5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1045291-C Therapeutic agents BOOTS CO PLC (GB) 1999-09-29 CN disclosed
EP-0618900-B1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS KNOLL AG (DE) 1997-03-12 EP disclosed
US-5519034-A ANALGESICS THE BOOTS COMPANY PLC (GB) 1996-05-21 US disclosed
CN-1096780-A Therapeutic agents containing novel tetrahydroisoquinoline compounds BOOTS CO PLC (GB) 1994-12-28 CN disclosed
EP-0618900-A1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS. BOOTS CO PLC (GB) 1994-10-12 EP disclosed
WO-1993013073-A1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS THE BOOTS COMPANY PLC (GB) 1993-07-08 WO disclosed