SCHEMBL8750856

SCHEMBL8750856

N#CNC(=NCCc1ccccc1Cl)c1cncc(NC(=O)c2ccccc2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
LMNA P02545 2/20 0.44
ALDH1A1 P00352 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
KDM4E B2RXH2 1/20 0.39
HSD17B10 Q99714 1/20 0.39
GRK2 P25098 1/20 0.39
GRK5 P34947 1/20 0.39
GRK3 P35626 1/20 0.39
BCAT2 O15382 1/20 0.39
NTRK1 P04629 1/20 0.38
SCN2A Q99250 1/20 0.38
SCN10A Q9Y5Y9 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
NAMPT P43490 1/20 0.37
KCNK3 O14649 2/20 0.37
KDR P35968 1/20 0.37
KCNK9 Q9NPC2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8750849 1.00 MAPT (0.44) MAPTSMN1; SMN2LMNAALDH1A1NPSR1
SCHEMBL8750752 0.86 FAAH (0.42) SMN1; SMN2ALDH1A1SCN2ASCN10ANPC1
SCHEMBL8750758 0.86 FAAH (0.42) SMN1; SMN2ALDH1A1SCN2ASCN10ANPC1
SCHEMBL8750733 0.84 HRH4 (0.37) ALDH1A1SCN2ASCN10ANAMPTKDR
SCHEMBL8750735 0.84 HRH4 (0.37) ALDH1A1SCN2ASCN10ANAMPTKDR
SCHEMBL8750815 0.83 HTR3E (0.38) SMN1; SMN2ALDH1A1NTRK1SCN2ASCN10A
SCHEMBL8750820 0.83 HTR3E (0.38) SMN1; SMN2ALDH1A1NTRK1SCN2ASCN10A
SCHEMBL8750851 0.83 GRK2 (0.36) ALDH1A1KDM4EGRK2NTRK1SCN2A
SCHEMBL8750847 0.83 GRK2 (0.36) ALDH1A1KDM4EGRK2NTRK1SCN2A
SCHEMBL8750772 0.83 HTR3E (0.38) ALDH1A1NTRK1SCN2ASCN10AKCNJ11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0634400-B1 PYRIDINECARBOXIMIDAMIDE COMPOUND AND USE THEREOF KIRIN BREWERY (JP) 1997-04-02 EP disclosed
US-5508293-A TREATING HYPERTENSION, ANGINA PECTORIS KIRIN BEER KABUSHIKI KAISHA (JP) 1996-04-16 US disclosed
EP-0634400-A1 PYRIDINECARBOXIMIDAMIDE COMPOUND AND USE THEREOF KIRIN BEER KABUSHIKI KAISHA (JP) 1995-01-18 EP disclosed