SCHEMBL8750992

SCHEMBL8750992

COC(=O)NCc1cccc(CNC(=O)O)c1

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.58
CYP1A2 P05177 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C9 P11712 1/20 0.54
CYP2C19 P33261 1/20 0.54
SMN1; SMN2 Q16637 3/20 0.51
ALDH1A1 P00352 4/20 0.50
KMT2A Q03164 2/20 0.48
ESR1 P03372 1/20 0.48
POLB P06746 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
HTT P42858 1/20 0.48
MMP13 P45452 1/20 0.48
MEN1 O00255 1/20 0.48
LMNA P02545 1/20 0.47
MAPT P10636 1/20 0.47
PKM P14618 1/20 0.47
ALOX12 P18054 1/20 0.47
HPGD P15428 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3895476 0.93 TSHR (0.66) TSHRSMN1; SMN2ALDH1A1KMT2AESR1
SCHEMBL8059189 0.87 CYP1A2 (0.68) TSHRCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL28540163 0.87 TSHR (0.61) TSHRCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL20457819 0.87 TSHR (0.66) TSHRCYP1A2CYP2C19SMN1; SMN2KMT2A
SCHEMBL8257957 0.86 TSHR (0.58) TSHRCYP2D6CYP2C19SMN1; SMN2ALDH1A1
SCHEMBL13450827 0.85 TSHR (0.57) TSHRCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL13037029 0.85 TSHR (0.57) TSHRCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL17863562 0.84 MMP13 (0.61) TSHRSMN1; SMN2ALDH1A1MMP13LMNA
SCHEMBL17346792 0.84 TSHR (0.53) TSHRSMN1; SMN2ALDH1A1KMT2AMEN1
SCHEMBL1720194 0.83 ALDH1A1 (0.67) TSHRCYP1A2CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0609786-B1 Process for producing urethane compound MITSUBISHI GAS CHEMICAL CO (JP) 1997-04-09 EP disclosed
US-5391805-A Process for producing urethane compound MITSUBISHI GAS CHEMICAL COMPANY INC. (JP) 1995-02-21 US disclosed
EP-0609786-A1 Process for producing urethane compound MITSUBISHI GAS CHEMICAL COMPANY, INC. (JP) 1994-08-10 EP disclosed
EP-0436800-B1 Process for producing isocyanate compound MITSUBISHI GAS CHEMICAL CO (JP) 1994-02-02 EP disclosed
US-5166414-A Process for producing isocyanate compound MITSUBISHI GAS CHEMICAL COMPANY, INC. (JP) 1992-11-24 US disclosed
EP-0436800-A1 Process for producing isocyanate compound MITSUBISHI GAS CHEMICAL COMPANY, INC. (JP) 1991-07-17 EP disclosed