SCHEMBL875438

SCHEMBL875438

CCCC(O)(O)Cc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2C9 P11712 1/20 0.48
SLC6A2 P23975 1/20 0.45
TAAR1 Q96RJ0 1/20 0.45
FDPS P14324 1/20 0.44
TP53 P04637 1/20 0.42
LMNA P02545 1/20 0.42
CYP2D6 P10635 1/20 0.42
TRPA1 O75762 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HIF1A Q16665 1/20 0.41
GAA P10253 1/20 0.40
ALOX12 P18054 1/20 0.40
ESR1 P03372 1/20 0.39
ESR2 Q92731 1/20 0.39
KCNA5 P22460 1/20 0.38
TSHR P16473 1/20 0.37
RIPK1 Q13546 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22289183 0.84 CSNK1E (0.45) CYP2C19CYP1A2CYP2C9TP53SMN1; SMN2
SCHEMBL28920634 0.84 CSNK1E (0.45) CYP2C19CYP1A2CYP2C9TP53SMN1; SMN2
SCHEMBL27671625 0.83 CYP2C19 (0.48) CYP2C19CYP1A2CYP2C9SLC6A2TAAR1
SCHEMBL9545396 0.83 CYP2C19 (0.48) CYP2C19CYP1A2CYP2C9SLC6A2TAAR1
SCHEMBL19030861 0.82 CYP1A2 (0.52) CYP2C19CYP1A2CYP2C9SLC6A2TAAR1
SCHEMBL10476772 0.81 CYP1A2 (0.61) CYP2C19CYP1A2CYP2C9SLC6A2TAAR1
SCHEMBL15255042 0.81 SLC6A2 (0.48) CYP2C19CYP1A2CYP2C9SLC6A2TAAR1
SCHEMBL8643657 0.79 SLC6A2 (0.52) CYP2C19CYP1A2CYP2C9SLC6A2TAAR1
SCHEMBL3401044 0.78 CYP1A2 (0.70) CYP2C19CYP1A2CYP2C9SLC6A2TAAR1
SCHEMBL2579939 0.77 CYP1A2 (0.52) CYP2C19CYP1A2CYP2C9SLC6A2TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9359306-B2 Process for preparing pan-CDK inhibitors of the formula (I), and intermediates in the preparation BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-06-07 US disclosed
US-20150118480-A1 LOW DENSITY EPOXY COMPOSITION WITH LOW WATER UPTAKE 3M INNOVATIVE PROPERTIES COMPANY 2015-04-30 US disclosed
EP-2653486-B1 Low density epoxy composition with low water uptake 3M INNOVATIVE PROPERTIES CO (US) 2014-12-03 EP disclosed
WO-2013158517-A1 LOW DENSITY EPOXY COMPOSITION WITH LOW WATER UPTAKE 3M INNOVATIVE PROPERTIES COMPANY (US) 2013-10-24 WO disclosed
EP-2653486-A1 Low density epoxy composition with low water uptake 3M Innovative Properties Company (US) 2013-10-23 EP disclosed
US-20130245261-A1 PROCESS FOR PREPARING PAN-CDK INHIBITORS OF THE FORMULA (I), AND INTERMEDIATES IN THE PREPARATION BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-09-19 US disclosed
EP-2619186-A1 PROCESS FOR PREPARING PAN-CDK INHIBITORS OF THE FORMULA (I), AND INTERMEDIATES IN THE PREPARATION Bayer Pharma Aktiengesellschaft (DE) 2013-07-31 EP disclosed
WO-2012038411-A1 PROCESS FOR PREPARING PAN-CDK INHIBITORS OF THE FORMULA (I), AND INTERMEDIATES IN THE PREPARATION BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-03-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130245261-A1 PROCESS FOR PREPARING PAN-CDK INHIBITORS OF THE FORMULA (I), AND INTERMEDIATES IN THE PREPARATION CDK1, CDK9, CDK6 CYP2C19 708/4885CYP1A2 1630/4885CYP2C9 1377/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.