SCHEMBL8763131

SCHEMBL8763131

C[C@H](NC(=O)c1c[nH]c(CCc2ccccc2)n1)C(=O)NC(C=O)CC(=O)O

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 15/20 0.47
IL1B P01584 2/20 0.42
CAPN1 P07384 1/20 0.39
LTA4H P09960 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL949786 1.00 CASP1 (0.47) CASP1IL1BCAPN1LTA4H
SCHEMBL949927 0.91 CASP1 (0.43) CASP1IL1BLTA4H
SCHEMBL27457960 0.91 CASP1 (0.43) CASP1IL1BLTA4H
SCHEMBL8762987 0.91 CASP1 (0.43) CASP1IL1BLTA4H
SCHEMBL8764720 0.89 PDE2A (0.39) CASP1IL1B
SCHEMBL949374 0.89 PDE2A (0.39) CASP1IL1B
SCHEMBL8763116 0.83 CASP1 (0.48) CASP1IL1BCAPN1LTA4H
SCHEMBL948289 0.83 CASP1 (0.48) CASP1IL1BCAPN1LTA4H
SCHEMBL12914534 0.81 MMP2 (0.52) CASP1IL1BCAPN1
SCHEMBL8764281 0.80 CASP1 (0.51) CASP1IL1BCAPN1LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0784628-A1 INHIBITORS OF INTERLEUKIN-1$g(b) CONVERTING ENZYME Vertex Pharmaceuticals Incorporated (US) 1997-07-23 EP disclosed
WO-1995035308-A1 INHIBITORS OF INTERLEUKIN-1β CONVERTING ENZYME VERTEX PHARMACEUTICALS INCORPORATED (US) 1995-12-28 WO disclosed